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CaMK Ca2+/calmodulin dependent kinase

Inhibitors

Cat.No.  Name Information
M21332 Calmidazolium chloride Calmidazolium chloride (R 24571) is a calmodulin antagonist that antagonizes CaM-dependent phosphodiesterase and calmodulin-induced activation of Ca2+-transporting ATPase in erythrocytes with IC50s of 0.15 and 0.35 μM, respectively. it is also used in anticancer studies. It binds CaMK with a Kd value of 3 nM.
M14559 Syntide 2 TFA Syntide 2 (TFA), a Ca2+- and calmodulin (CaM)-dependent protein kinase II (CaMKII) substrate peptide, selectively inhibits the gibberellin (GA) response, leaving constitutive and abscisic acid-regulated events unaffected.
M14558 KN-93 phosphate KN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM.
M14557 CaMKII-IN-1 CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC.
M14556 Autocamtide-2-related inhibitory peptide TFA Autocamtide-2-related inhibitory peptide (TFA) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
M9624 KN-93 hydrochloride KN-93 hydrochloride is a cell-permeable inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMK-II) with a Ki of 370 nM.
M9266 STO-609 acetate STO-609 acetate is a cell-permeable inhibitor of calcium/calmodulin-dependent kinase kinases (CaMKK) isoforms CaMKKα and CaMKKβ with Ki of 80 and 15 ng/ml, respectively.
M9254 KN-92 phosphate KN-92 is an inactive analog of the CaM kinase II inhibitor KN-93.
M7481 W-7 hydrochloride W-7 Hydrochloride is a selective calmodulin antagonist. W-7 Hydrochloride inhibits Ca2+ -calmodulin-dependent phosphodiesterase and Myosin light chain kinase. The IC50 values were 28 μM and 51 μM, respectively. W-7 Hydrochloride can induce apoptosis and has anti-cancer activity.
M6868 KN 93 KN 93 is a caM kinase II inhibitor; also K + channel blocker (K V).
M3866 KN-92 KN-92 is an inactive analog of the CaM kinase II inhibitor KN-93.
M3623 A23187 A23187 is a calcium ionophore that induces Ca2+-dependent cell death by increasing intracellular calcium concentration.
M1928 KN-62 KN-62 is a selective, cell permeable inhibitor of calcium/calmodulin-dependent kinase II (CaMKII; IC50 = 900 nM).



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