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Abmole Inhibitor Catalog 2017

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Inhibitors

Cat.No.  Name Information
M9613 4-P-PDOT 4-P-PDOT is a MT2-receptor-specific antagonist, it is >300-fold more selective for MT2 than MT1.
M9611 S-Adenosylhomocysteine S-Adenosylhomocysteine, an intermediate in the synthesis of cysteine and adenosine, is an inhibitor for METTL3-METTL14 heterodimer complex (METTL3-14) with an IC50 of 0.9 µM.
M9609 SP-13786 SP-13786 (UAMC-1110) is a novel potent and selective inhibitor of fibroblast activation protein (fap), displaying low nanomolar inhibitory potency and high selectivity against the related dipeptidyl peptidases (dpps) dppiv, dpp9, dppii, and prolyl oligopeptidase (prep).
M9608 APX-115 APX-115 is a potent, orally active inhibitor of pan NADPH oxidase (Nox) with Ki of 1.08 μM, 0.57 μM, and 0.63 μM for Nox1, Nox2 and Nox4, respectively.
M9607 VU0119498 VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM).
M9606 VU0238441 VU0238441 is a potent agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
M9599 NB-598 NB-598 is a potent competitive inhibitor of squalene epoxidase (SE).
M9595 Upamostat Upamostat is an orally bioavailable, second generation serine protease inhibitor targeting the human urokinase plasminogen activator (uPA) system with potential antineoplastic and antimetastatic activities.
M9594 EDC.HCl Crosslinker EDC.HCl Crosslinker is a zero-length crosslinker that can be used to conjugate carboxyl functional groups to primary amines.
M9593 Iminodiacetic acid Iminodiacetic acid is a bovine liver glutamate dehydrogenase inhibitor.
M9591 D-(+)-Trehalose dihydrate D-(+)-Trehalose dihydrate is used as a food ingredient and pharmaceutical excipient.
M9583 Dansylsarcosine piperidinium salt Dansylsarcosine piperidinium salt
M9582 Tris Dodecyl Sulfate Tris Dodecyl Sulfate
M9580 β-Nicotinamide mononucleotide β-nicotinamide mononucleotide (β-NM) is an intermediate in NAD+ biosynthesis produced from nicotinamide (NAM) and phosphoribosyl pyrophosphate (PRPP) by nicotinamide phosphoribosyl transferase enzyme with no toxicity.
M9579 XMD-17-51 XMD-17-51 is a potent and selective NUAK1 inhibitor.
M9572 α-Melanocyte stimulating hormone α-Melanocyte-stimulating hormone (α-MSH) is a tridecapeptide, mostly produced by the cells in the brain, pituitary and circulation.
M9571 Pin1 inhibitor API-1 Pin1 inhibitor API-1 is a Pin1 inhibitor with an IC50 of 72.3 nM.
M9568 SC-26196 SC-26196 is a potent, orally active D6D inhibitor (IC50 = 0.2 µM in a rat liver microsomal assay) that completely blocks the conversion of linoleic acid to arachidonic acid (AA).
M9567 Leptin (116-130) mouse Leptin (116-130) mouse is a synthetic leptin peptide fragment.
M9564 Lumiflavine Lumiflavine is a structural analog of the water-soluble vitamin riboflavin.
M9563 2,1,3-Benzothiadiazole-5-carbaldehyde 2,1,3-Benzothiadiazole-5-carbaldehyde
M9560 Paquinimod Paquinimod is a S100A9 inhibitor preventing S100A9 binding to TLR-4.
M9557 BAY-1816032 BAY-1816032 is a potent and oral available BUB1 (budding uninhibited by benzimidazoles 1) kinase inhibitor with an IC50 of 7 nM.
M9556 Potassium thiocyanate Potassium thiocyanate is an inorganic potassium salt. Potassium thiocyanate (KSCN) may be used for the colorimetric quantification of intracellular iron content of the superparamagnetic iron oxide (SPIO) nanoparticles.
M9552 Stigmasterol Stigmasterol is a plant sterol which has been focused on the cholesterol-lowering activity and is valued as an anti-stiffness factor in the therapy of rheumatic diseases.
M9549 Nonaethylene glycol monododecyl ether Nonaethylene glycol monododecyl ether is a nonionic surfactant and polyethylene glycol (PEG) detergent that can be used to form initial coalesced O/W emulsion droplets, as well as for protein separation and purification.
M9544 Heparan Sulfate Heparan sulfate is a complex and linear polysaccharide, which expressed abundantly on the cell surface and in the extracellular matrix.
M9543 Dextran Dextran (Dextran 40) has an inhibitory effect on thrombocyte aggregation.
M9537 Protein kinase inhibitors 1 Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
M9536 VBIT-12 VBIT-12 is a potent inhibitor of VDAC1, directly interacting with purified VDAC1 and reducing its channel conductance.
M9531 NADP disodium salt NADP disodium salt is a participant coenzyme in aerobic and anaerobic oxidations.
M9529 L-Glutamic acid monosodium salt hydrate L-Glutamic acid monosodium salt hydrate is also a Kainate receptor, NMDA receptor and quisqualate receptor agonist; an excitatory amino acid neurotransmitter.
M9524 Lipopolysaccharides Lipopolysaccharides (LPS) is an endotoxin derived from the outer leaflet of the outer membrane of Gram-negative bacteria.
M9523 PEG6000 PEG6000 is a neutral and biocompatible hydrophilic polymer.
M9517 Sodium hippurate Hippuric acid is a low molecular weight phenolic carboxylic acid urinary metabolite that may be a useful urinary biomarker for certain cancers such as gastric cancer and oxidative stress.
M9511 DO264 DO264 is a potent selective, and in vivo active ABHD12 inhibitor, with an IC50 of 11 nM.
M9507 ML-109 ML-109 is a full agonist of TSHR (thyroid stimulating hormone receptor) with an EC50 of 40 nM.
M9504 D-Desthiobiotin D-Desthiobiotin is a biotin derivative used in affinity chromatography and protein chromatography, also can be used for protein and cell labeling, detection and isolation.
M9502 CVT-12012 CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhibitor, with IC50s of 38 nM, 6.1 nM for rat microsomal and human HEPG2, respectively.
M9499 TH-257 TH-257 is a potent and selective allosteric LIMK 1/2 inhibitor with IC50 values of 84 nM and 39 nM, respectively.
M9498 CADD522 CADD522 is a novel small molecule inhibitor of RUNX2, downregulates RUNX2-mediated transcription of downstream target genes by inhibiting RUNX2-DNA binding, with an IC50 of 10 nM.
M9497 ML-792 ML-792 is a potent and selective SAE inhibitor with nanomolar potency in cellular assays.
M9495 FGH10019 FGH10019 is a novel SREBP (sterol regulatory element-binding protein) inhibitor, with IC50 of 1 μM.
M9483 Azeliragon Azeliragon is a potent and orally active RAGE inhibitor.
M9481 ML092 ML092 (Cruzain-IN-1) is a selective, covalent and reversible Cruzain inhibitor, with IC50 of 10 nM.
M9479 YHO-13177 YHO-13177 is a potent and specific inhibitor of breast cancer resistance protein (BCRP/ABCG2).
M9477 NSC348884 NSC348884 is a nucleophosmin inhibitor, inhibits cell proliferation at an IC50 of 1.7-4.0 μM in distinct cancer cell lines.
M9475 Sardomozide dihydrochloride Sardomozide dihydrochloride (also known as SAM486A or CGP48664) is a second-generation polyamine synthesis inhibitor, which inhibits the activity of the polyamine biosynthetic enzyme S-adenosylmethionine decarboxylase (SAMDC).
M9472 Hydroxyhexamide Hydroxyhexamide is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agents.
M9470 Aftin-4 Aftin-4 is an inducer of Aß-42 peptide production.


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