Catalog

Others Others

Inhibitors

Cat.No.	Name	Information
M9089	SAR7334	SAR7334 is a novel, highly potent and bioavailable inhibitor of TRPC6 channels.
M9087	FICZ	FICZ is a potent aryl hydrogen receptor (AhR) agonist.
M9086	NAD+	NAD+ is a coenzyme composed of ribosylnicotinamide 5'-diphosphate coupled to adenosine 5'-phosphate by pyrophosphate linkage.
M9084	STING-Inducer-1	STING-Inducer-1 (ML RR-S2 CDA) is an inducer of STING (stimulator of interferon genes).
M9082	ISO-1	ISO-1, also known as MIF Antagonist, is a MIF inhibitor with an IC50 of 7 uM.
M9081	Sodium Stibogluconate	Sodium Stibogluconate is a potent inhibitor of protein tyrosine phosphatase.
M9076	NADPH tetrasodium salt	NADPH tetrasodium salt is a cofactor, used to donate electrons and a hydrogens to reactions catalyzed by some enzymes.
M9075	(R)-(+)-Etomoxir sodium salt	(R)-(+)-Etomoxir sodium salt is the R-form of Etomoxir sodium salt.
M9072	ATP	Adenosine triphosphate (ATP) is an adenine nucleotide containing three phosphate groups esterified to the sugar moiety.
M9071	Amyloid beta-peptide(25-35)	Amyloid beta-peptide(25-35) is the fragment Aβ(25-35) of the Alzheimer's amyloid β-peptide, has shown neurotoxic activities in cultured cells.
M9068	Mitoquinone mesylate	Mitoquinone mesylate is a TPP-based, mitochondrially targeted antioxidant.
M9064	Oxytocin acetate	Oxytocin acetate is a mammalian neurohypophysial hormone.
M9063	TLR2-IN-C29	TLR2-IN-C29 is an inhibitor of TLR2/1 and TLR2/6 signaling.
M9062	Necrosulfonamide	Necrosulfonamide is an MLKL inhibitor with IC50 value of 124 nM in human HT-29.
M9060	RSL3	RSL3 is an inhibitor of the glutathione (GSH) peroxidase 4, which can inhibit the cysteine/glutamate amino acid transporter system.
M9058	Varenicline hydrochloride	Varenicline hydrochloride is a nicotinic receptor partial agonist.
M9057	XMU-MP-1	XMU-MP-1 is a potent and selective MST1/2 inhibitor with IC50 values of 71.1 ± 12.9 nM and 38.1 ± 6.9 nM, respectively.
M9053	D-Luciferin	D-Luciferin is a light-emitting compound, also a natural substrate of luciferases.
M9052	ST2825	ST-2825 is MyD88 inhibitor.
M9051	FCCP	FCCP is a mitochondrial uncoupling agent.
M9049	MPTP HCl	MPTP hcl is a compound to the neurotoxin MPP+ which causes permanent symptoms of Parkinson's disease.
M9048	Etomoxir	Etomoxir is a potent inhibitor of carnitine palmitoyltransferase-I (CPT-1).
M9043	INCB057643	INCB057643 is a novel BET inhibitor.
M9038	Photochlor	Photochlor is a lipophilic, second-generation, chlorin-based photosensitizer.
M9037	AMPPD	AMPPD is a new biochemistry ultrasensitive alkaline phosphatase substrate.
M9036	DM1-SMCC	DM1-SMCC is DM1 with a reactive linker SMCC, which can react with antibody to make ADC.
M9034	Mitapivat	Mitapivat is a potent human R-type pyruvate kinase (PKR) inhibitor.
M9033	VH-298	VH-298 is a potent VHL inhibitor that stabilizes HIF-α and elicits a hypoxic response via a different mechanism, with a Kd value of 80 to 90 nM.
M9031	6-Methylcoumarin	6-Methylcoumarin belongs to the class of organic compounds known as coumarins and derivatives.
M9021	BTTAA	BTTAA is a Cu(I)-stabilizing ligand, whch performs potently with ubiquitin Glu18AzF.
M9016	Ezutromid	Ezutromid (also known as BMN-195 and SMT C1100) is a first orally bioavailable utrophin's translation modulator with EC50 of 0.4 uM.
M9015	GNE-495	GNE-495 is a potent and selective MAP4K4 inhibitor with an IC50 of 3.7 nM.
M9002	ML281	ML-281 is a potent ans selective STK33 inhibitor with IC50 value of 14 nM.
M9001	ML-265	ML-265 (TEPP-46) is a potent and selective activator of recombinant pyruvate kinase M2 (PKM2).
M8990	LB-100	LB-100 is a water soluble protein phosphatase 2A (PP2A) inhibitor, with IC50 of 0.85 μM and 3.87 μM in BxPc-3 and Panc-1 cells.
M8984	Denosumab	Denosumab is designed to target RANKL (RANK ligand), a protein that acts as the primary signal to promote bone removal/resorption.
M8983	Compstatin	Compstatinis is a 13-residue cyclic peptide, binds to complement component C3 and inhibits complement activation with IC50 of 12 μM.
M8982	Azaserine	Azaserine is an inhibitor of the rate limiting step of the hexosamine biosynthethic pathway (HBP) and an irreversible inhibitor of GGT1 (gamma-Glutamyltranspeptidase).
M8979	TM6008	TM6008 is a novel PHD inhibitor, which inhibited PHD and stabilized HIF activity in vitro.
M8976	ASP9521	ASP9521 is a novel, selective, orally bioavailable inhibitor of 17β-hydroxysteroid dehydrogenase type 5 (17βHSD5; AKR1C3).
M8974	ALW-II-41-27	ALW-II-41-27 is a Eph receptor tyrosine kinase inhibitor with an IC50 of 11 nM for EPHA2.
M8968	FPS-ZM1	FPS-ZM1 is a high-affinity RAGE-specific blocker that inhibits amyloid-β binding to RAGE with a Ki of 25 nM.
M8965	2,6-Diaminopurine	2,6-Diaminopurine is a compound used to treat leukemia.
M8964	Thymidine	Thymidine is a pyrimidine nucleoside that is composed of the pyrimidine base thymine attached to the sugar deoxyribose.
M8960	LY2334737	LY2334737 is an orally available valproic acid ester of gemcitabine, a broad-spectrum antimetabolite with antineoplastic activity.
M8948	TUG-891	TUG-891 is a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120).
M8943	GSK2981278	GSK2981278 is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).
M8935	EXP-3174	EXP-3174 is a potent AT1 antagonist with Kis of 0.57 and 0.67 nM for rat and human forms, respectively.
M8929	NAV-2729	NAV-2729 is a selective ARF6 inhibitor with IC50 value of 1.0 μM.
M8922	Brevianamide F	Brevianamide F belongs to a class of naturally occurring 2,5-diketopiperazines.

Signaling Pathways

Product Type

Others Others

Get to Know Us

Customer Support

Resources

Contact Us