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Inhibitors

Cat.No.	Name	Information
M8990	LB-100	LB-100 is a water soluble protein phosphatase 2A (PP2A) inhibitor, with IC50 of 0.85 μM and 3.87 μM in BxPc-3 and Panc-1 cells.
M8984	Denosumab	Denosumab is designed to target RANKL (RANK ligand), a protein that acts as the primary signal to promote bone removal/resorption.
M8983	Compstatin	Compstatinis is a 13-residue cyclic peptide, binds to complement component C3 and inhibits complement activation with IC50 of 12 μM.
M8982	Azaserine	Azaserine is an inhibitor of the rate limiting step of the hexosamine biosynthethic pathway (HBP) and an irreversible inhibitor of GGT1 (gamma-Glutamyltranspeptidase).
M8979	TM6008	TM6008 is a novel PHD inhibitor, which inhibited PHD and stabilized HIF activity in vitro.
M8976	ASP9521	ASP9521 is a novel, selective, orally bioavailable inhibitor of 17β-hydroxysteroid dehydrogenase type 5 (17βHSD5; AKR1C3).
M8974	ALW-II-41-27	ALW-II-41-27 is a Eph receptor tyrosine kinase inhibitor with an IC50 of 11 nM for EPHA2.
M8968	FPS-ZM1	FPS-ZM1 is a high-affinity RAGE-specific blocker that inhibits amyloid-β binding to RAGE with a Ki of 25 nM.
M8965	2,6-Diaminopurine	2,6-Diaminopurine is a compound used to treat leukemia.
M8964	Thymidine	Thymidine is a pyrimidine nucleoside that is composed of the pyrimidine base thymine attached to the sugar deoxyribose.
M8960	LY2334737	LY2334737 is an orally available valproic acid ester of gemcitabine, a broad-spectrum antimetabolite with antineoplastic activity.
M8948	TUG-891	TUG-891 is a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120).
M8943	GSK2981278	GSK2981278 is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).
M8935	EXP-3174	EXP-3174 is a potent AT1 antagonist with Kis of 0.57 and 0.67 nM for rat and human forms, respectively.
M8929	NAV-2729	NAV-2729 is a selective ARF6 inhibitor with IC50 value of 1.0 μM.
M8922	Brevianamide F	Brevianamide F belongs to a class of naturally occurring 2,5-diketopiperazines.
M8913	Telotristat ethyl	Telotristat ethyl, also known as LX1606, is an oral serotonin synthesis inhibitor or peripheral tryptophan hydroxylase (TPH) inhibitor.
M8912	ML-18	ML18 is Bombesin receptor subtype 3 (BRS-3) antagonist (IC50 = 4.8 μM).
M8907	Acecainide HCl	Acecainide HCl, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide.
M8906	Sematilide hydrochloride	Sematilide (CK-1752) hydrochloride is a novel class III antiarrhythmic agent.
M8905	EBE-A22	EBE-A22 is a derivative of PD 153035, has no effect on EGF-R TK but maintains a high cytotoxic profile.
M8904	NIH-12848	NIH-12848 is a putative phosphatidylinositol 5-phosphate 4-kinase γ (PI5P4Kγ) inhibitor.
M8901	CHS-828	CHS-828 (GMX1778) is a potent and specific inhibitor of NAMPT with IC50 and Kd value of <25 nM and 120 nM, respectively.
M8898	APY0201	APY0201 is a potent and selective IL-12/23 inhibitor.
M8896	MDK36122	MDK36122, also known as H-PGDS Inhibitor I, is a Prostaglandin D Synthase (hematopoietic-type) Inhibitor with an IC50 Value of 0.7 nM.
M8894	GJ-103	GJ-103 is an active analog of the read-through compound GJ072.
M8893	Miriplatin	Miriplatin is a chemotherapy agent which belongs to the class of alkylating agents.
M8892	Coluracetam	Coluracetam (MKC-231) is a new choline uptake enhancer.
M8891	AI-1	AI-1 is a negative regulator of Nrf2.
M8890	Forchlorfenuron	Forchlorfenuron is a synthetic cytokinin that inhibits septins and exhibits anti-parasitic, anticancer, and anti-angiogenic activities.
M8889	6-Methoxy-2-naphthoic acid	6-Methoxy-2-naphthoic acid is an NMDA receptor modulator.
M8884	Febantel	Febantel is a veteran anthelmintic (wormer) compound belonging to the chemical class of the benzimidazoles.
M8883	Ceforanide	Ceforanide is a new cephalosporin with antibacterial activity and has a longer elimination half-life than any currently available cephalosporin.
M8878	Inositol Nicotinate	Inositol Nicotinate is a formulation of niacin, which is also called vitamin B3, an essential human nutrient.
M8875	ND-630	ND-630 is an ACC inhibitor of human ACC1 and ACC2 with IC50 values of 2.1 and 6.1 nM, respectively.
M8873	D-Luciferin potassium salt	D-Luciferin potassium salt is the substrate of luciferases that catalyze the production of light in bioluminescent insects.
M8872	ZD 7114 hydrochloride	ZD 7114 is a selective β3 adrenergic receptor agonist.
M8870	Zopolrestat	Zopolrestat is an inhibitor of Aldose Reductase.
M8869	Zinterol hydrochloride	Zinterol Hydrochloride is a β2 adrenergic receptor selective agonist.
M8868	Zerumbone	Zerumbone is a TRAIL-induced apoptosis potentiator.
M8867	Zaragozic acid A trisodium salt	Potent inhibitor, in vivo and in vitro, of mammalian, fungal and Saccharomyces cervisiae squalene synthase.
M8866	Zonisamide sodium salt	Zonisamide sodium salt is an anti-epileptic.
M8865	Zimelidine dihydrochloride	Serotonin transport blocker; antidepressant.
M8864	Zotepine	Zotepine is an atypical antipsychotic.
M8863	YM 976	Phosphodiesterase type IV (PDE4) inhibitor.
M8862	YH439	YH439 is an aryl hydrocarbon receptor activator.
M8861	Xaliproden hydrochloride	5-HT_1A serotonin receptor agonist; neuroprotectant.
M8860	X80	X80 is an inhibitor of xeroderma pigmentosum group A protein (XPA protein) required for the removal of all types of DNA lesions repaired by nucleotide excision repair Including both transcription coupled and global genomic nucleotide excision repair.
M8859	Xestospongin C	Xestospongin C is a selective, reversible and membrane-permeable inhibitor of IP₃ receptor.
M8858	XE-991	XE-991 is a KCNQ channel blocker; which is more potent than linopiridine.

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