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Abmole Inhibitor Catalog 2017

GPR G protein-coupled receptor


Cat.No.  Name Information
M5292 GPR120-IN-1 GPR120-IN-1是选择性的Gpr120激动剂,logEC50值为?7.62。
M5187 GSK137647A GSK137647A is a selective FFA4 agonist for human, Mouse and Rat FFA4 with pEC50 values of 6.3, 6.2 and 6.1, respectively.
M3773 PSN-375963 PSN375963 is a potent and selective agonist of GPR119 that shows similar potency to oleoyl ethanolamide (OEA) at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 8.4 and 7.9 µM, respectively (EC50 values for OEA are 3.2 and 2.9 µM, respectively).
M3771 PSN632408 PSN632408 is a novel, selective and small-molecule agonist of human and mouse GPR119 with EC50 values of 5.6±0.99 μM and 7.9±0.7 μM, respectively.
M3766 AR-231453 AR-231453 is a potent, selective G-protein coupled receptor 119 (GPR119) agonist (EC50 = 0.68 nM).
M3632 MBX-2982 MBX-2982 is a selective, orally-available GPR119 agonist for the treatment of type 2 diabetes.
M3321 GSK1292263 GSK1292263 is a novel GPR119 agonist, showing potential for the treatment of type 2 diabetes.
M2418 AZD1981 AZD1981 is a potent, selective CRTh2 (DP2) receptor antagonist with IC50 of 4 nM, showing >1000-fold selectivity over more than 340 other enzymes and receptors, including DP1.
M2384 AMG-837 AMG 837 is a potent, orally bioavailable GPR40 agonist with EC50 of 14 nM.
M2091 OC000459 OC000459 is a potent, selective, and orally active D prostanoid receptor 2 antagonist.
M2054 TAK-875 TAK-875 is a novel, orally available, selective GPR40 agonist.
M2020 GW9508 GW9508 is a small-molecule agonist of the fatty acid receptors GPR40 and GPR120.

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