Inhibitor/Activator
| Cat.No. | Name | Information |
|---|---|---|
| M53099 | Neuropeptide EI, rat | Neuropeptide EI, rat displays functional melanin concentrating hormone (MCH)-antagonist and melanocyte-stimulating hormone (MSH) agonist activity in different behavioral paradigms. |
| M53098 | (Phe13, Tyr19)-MCH (human, mouse, rat) | (Phe13,Tyr19)-MCH (human, mouse, rat) is a potent SLC-1 and S643b receptor ligand. |
| M53097 | Melanin Concentrating Hormone, salmon | Melanin Concentrating Hormone, salmon is a 19-amino-acid neuropeptide initially identified in the pituitary gland of teleost fish, which regulates food intake, energy balance, sleep state, and the cardiovascular system. |
| M53096 | MCH(human, mouse, rat) | MCH (human, mouse, rat) is a potent peptide agonist of MCH-R and exhibits binding IC50 values of 0.3nM and 1.5 nM for MCH1R and MCH2R, respectively. |
| M53095 | Ac-hMCH(6-16)-NH2 | Ac-hMCH(6-16)-NH2 binds to and activates equally well both human MCH receptors present in the brain (non-selective agonist), with IC50 values of 0.16 nM and 2.7 nM for MCH-1R and MCH-2R. |
| M49639 | ML192 | ML192 is a selective ligand antagonist of GPR55. |
| M49445 | BAY-3178275 | BAY-3178275 is an antagonist targeting GPR84 for studies related to diabetic neuropathic pain. |
| M45123 | GSK256073 | GSK256073 is a potent, selective, orally active GPR109A agonist and a potent and persistent HCA2 agonist with a pEC50 of 7.5 (Human HCA2). In addition, GSK256073 significantly improves glucose homeostasis by inhibiting lipid degradation and has potential for the study of type 2 diabetes mellitus (T2DM) and dyslipidemia. |
| M45110 | GSK4381406 | GSK4381406 is a first-in-class, orally active GPR35 agonist for studies related to inflammatory bowel disease (IBD). |
| M43816 | EVO756 | EVO756 is a Mas-related G protein-coupled receptor X2 (MRGPRX2) antagonist that can be used in studies related to urticaria. |
| M43815 | EP262 | EP262 is an orally active small molecule antagonist of the Mas-related G protein-coupled receptor (MRGPRX2) for studies related to mast cell-mediated diseases such as chronic urticaria and atopic dermatitis. |
| M41868 | hMCH-1R antagonist 1 | hMCH-1R antagonist 1 is an effective and selective antagonist of human melanin-concentrating hormone receptor 1 (hMCHR1) with an KB value of 3.6 nM. |
| M41851 | Kisspeptin 234 | Kisspeptin 234, is a 10 amino acid peptide as well as a kisspeptin receptor (KISS1, GPR54) antagonist. |
| M41850 | Kisspeptin 234 TFA | Kisspeptin 234 TFA, is a 10 amino acid peptide as well as a kisspeptin receptor (KISS1, GPR54) antagonist. |
| M41842 | Bufrolin | Bufrolin is a Cromoglycate (histamine release inhibitor) analog and a high potency agonist of GPR35. |
| M41841 | GPR119 agonist 2 | GPR119 agonist 2 is an orally active GPR119 agonist. |
| M41840 | GPCR agonist-2 | GPCR agonist-2 is a GPCR GPR109b (HM74) agonist, with a pEC50 value of 6.51. |
| M41821 | AM-5262 | AM-5262 is a GPR40 full agonist with an EC50 value of 0.081 μM. |
| M38958 | (±)-Pinocembrin | (±)-Pinocembrin ((±)-5,7-Dihydroxyflavanone) is a GPR120 ligand able to promote wound healing in HaCaT cell line. |
| M31033 | BAM(8-22) TFA | BAM(8-22) TFA, a proteolytically cleaved product of proenkephalin A, is a potent activator of Mas-related G-protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces scratching in mice in an Mrgpr-dependent manner. |
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