Free shipping on all orders over $ 500
  Catalog
Abmole Inhibitor Catalog 2017

Endothelin Receptor Endothelin Receptor

Inhibitors

Cat.No.  Name Information
M5135 Ro-46-2005 Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM.
M2467 Bosentan Bosentan is an endothelin (ET) receptor antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively.
M2278 Bosentan Hydrate Bosentan is an endothelin (ET) receptors antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively.
M2205 Macitentan Macitentan is an orally-active, tissue-targeting dual ET receptor antagonist.
M2029 Sitaxsentan sodium Sitaxsentan (TBC-11251) is an orally active, highly selective antagonist of endothelin A receptors.
M1951 Ambrisentan Ambrisentan is an orally active, highly selective antagonist of the endothelin-1 type A receptor.
M1816 Zibotentan Zibotentan (ZD4054) is a more selective and specific endothelin-A receptor (ETAR) antagonist with an IC50 value of 21 nM.


Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2017 AbMole BioScience. All Rights Reserved.