Inhibitors
Cat.No. | Name | Information |
---|---|---|
M9792 | Sarafotoxin S6c | Sarafotoxin S6c is a highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively). |
M9555 | Endothelin-1 (human, porcine) | Endothelin-1 (human, porcine) is a synthetic peptide with the sequence of human and swine Endothelin 1, which is a potent endogenous vasoconstrictor. |
M9554 | BQ-123 | BQ-123 is a selective endothelin A receptors (ETAR) antagonist with an IC50 value of 7.3 nM. |
M5135 | Ro-46-2005 | Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM. |
M2467 | Bosentan | Bosentan is an endothelin (ET) receptor antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively. |
M2278 | Bosentan Hydrate | Bosentan is an endothelin (ET) receptors antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively. |
M2205 | Macitentan | Macitentan is an orally-active, tissue-targeting dual ET receptor antagonist. |
M2029 | Sitaxsentan sodium | Sitaxsentan (TBC-11251) is an orally active, highly selective antagonist of endothelin A receptors. |
M1951 | Ambrisentan | Ambrisentan is an orally active, highly selective antagonist of the endothelin-1 type A receptor. |
M1816 | Zibotentan | Zibotentan (ZD4054) is a more selective and specific endothelin-A receptor (ETAR) antagonist with an IC50 value of 21 nM. |
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