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Abmole Inhibitor Catalog 2017

Dopamine Receptor Dopamine Receptor


Cat.No.  Name Information
M9601 Cariprazine Cariprazine is a D2 and D3 receptor partial agonist, with high selectivity towards the D3 receptor.
M9482 PD-168077 maleate PD-168077 maleate is a potent D4 dopamine receptor agonist (Ki = 8.7 nM), with > 400-fold and > 300-fold selectivity over D2 / D3 subtypes, respectively.
M9099 SCH23390 SCH23390 is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types, respectively).
M9049 MPTP HCl MPTP hcl is a compound to the neurotoxin MPP+ which causes permanent symptoms of Parkinson's disease.
M9022 SKF38393 HCl SKF38393 HCl is a selective D1 dopamine receptor agonist with IC50 of 110 nM.
M7832 6-Hydroxydopamine hydrochloride 6-Hydroxydopamine hydrochloride is an antagonist of the neurotransmitter dopamine.
M7279 SCH 23390 hydrochloride SCH 23390 hydrochloride is a standard selective D 1-like antagonist; also 5-HT 2C and 5-HT 1C agonist and K ir3 channel blocker.
M5984 Sulpiride Sulpiride is a dopamine D2-receptor antagonist. It has been used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.
M5914 rac-Rotigotine (Hydrochloride) rac-Rotigotine Hcl is a high potency and selectivity agonist for D-2 receptor with Ki of 0.69 nM.
M5903 Promazine HCl Promazine (hydrochloride) is a D2 dopamine receptor antagonist, belongs to the phenothiazine class of antipsychotics, used to treat schizophrenia.
M5900 Prochlorperazine dimaleate salt Prochlorperazine dimaleate is a dopamine (D2) receptor antagonist.
M5891 Pramipexole dihydrochloride Pramipexole 2Hcl is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively.
M5872 Perphenazine Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
M5854 SB 277011 Hydrochloride Ligands acting as DRD3 antagonists (SB 277011-A) has shown some promise for reducing the influence of drug-associated cues on motivational behaviour.
M5848 Paliperidone Paliperidone, the main active metabolite of Risperidone, is a potent serotonin-2A and dopamine-2 receptor antagonist, used in the treatment of schizophrenia.
M5796 Molindone HCl Molindone is a therapeutic antipsychotic, used in the treatment of schizophrenia, works by blocking the effects of dopamine in the brain, leading to diminished psychoses.
M5739 Levosulpiride Levosulpiride is a selective antagonist for D2 dopamine receptors used as an antipsychotic and prokinetic agent.
M5686 Haloperidol Haloperidol is a potent dopamine D2 receptor antagonist.
M5642 Fenoldopam mesylate Fenoldopam is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation.
M5590 Dopamine HCl Dopamine HCl is a catecholamine neurotransmitter present in a wide variety of animals,And a dopamine D1-5 receptors agonist.
M5525 Clebopride malate Clebopride malate is a dopamine antagonist drug with antiemetic and prokinetic properties used to treat functional gastrointestinal disorders.
M5467 Brexpiprazole Brexpiprazole is a novel D2 dopamine and serotonin 1A partial agonist, called serotonin-dopamine activity modulator (SDAM), and a potent antagonist of serotonin 2A receptors, noradrenergic alpha 1B and 2C receptors.
M5410 Amisulpride Amisulpride is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.
M5350 (+,-)-Octopamine Octopamine (OA), a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates.
M5198 Fluphenazine dihydrochloride Fluphenazine dihydrochloride is a phenothiazine-class D1DR and D2DR inhibitor.
M4942 Metoclopramide hydrochloride hydrate Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic.
M3785 Flupenthixol dihydrochloride Flupenthixol dihydrochloride is a dopamine receptor antagonist which acts as a Neuroleptic agent as well as an antipsychotic.
M3675 Rotigotine Rotigotine is dopamine D2 and D3 receptor agonist with Ki values of 13 and 0.71 nM for D2 and D3 respectively.
M3674 Metoclopramide Metoclopramide is a dopamine D2 antagonist that is used as an antiemetic.
M3586 Pramipexole dihydrochloride Monohydrate Pramipexole dihydrochloride Monohydrate is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM.
M3338 Domperidone Domperidone is a dopamine blocker and an antidopaminergic reagent.
M3287 PD128907 hydrochloride PD 128907 hydrochloride is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.
M3250 Vanoxerine Vanoxerine (GBR-12909) is a potent and selective dopamine receptor inhibitor.
M3246 Amfebutamone hydrochloride Amfebutamone hydrochloride is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrine, respectively
M3242 Sumanirole Maleate Sumanirole maleate is a highly selective dopamine D2 receptor agonist with binding affinity of 9 nM and EC50 of about 46 nM, exhibits >200-fold selectivity over the other dopamine receptor subtypes.
M3165 Prochlorperazine dimaleate Prochlorperazine dimaleate is a D2 dopamine receptor antagonist.
M3088 Triflupromazine hydrochloride Triflupromazine is a member of a class of compounds called phenthiazines, which are dopamine D1/D2 receptor antagonists.
M3087 Trifluoperazine dihydrochloride Trifluoperazine is a dopamine D2 receptor inhibitor with IC50 of 1.1 nM.
M2987 Ropinirole hydrochloride Ropinirole a selective dopamine D2 receptors inhibitor with IC50 of 29 nM.
M2936 Phenothiazine Phenothiazine is a dopamine-2 (D2) receptor antagonist therefore decreases the effect of dopamine in the brain.
M2494 Cariprazine hydrochloride Cariprazine hydrochloride is a dopamine D3-receptor-preferring partial agonist that exhibits high selectivity and affinity to dopamine D3 and D2(L/S) receptors with pKi 10.07 and 9.16/9.31, respectively.
M1910 Nepicastat hydrochloride Nepicastat hydrochloride is a potent and selective inhibitor of both bovine and human dopamine-β-hydroxylase with IC50 of 8.5 nM and 9 nM, respectively.

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