Free shipping on all orders over $ 500
Abmole Inhibitor Catalog 2017

Calcium Channel Calcium Channel


Cat.No.  Name Information
M10363 Cyclic ADP-​ribose ammonium Cyclic ADP-ribose is a cyclic purine nucleotide that is synthesised from NAD+ by ADP-ribosyl cyclase; acts as an agonist at ryanodine receptors.
M9794 Ebselen Ebselen (SPI-1005) is a potent voltage-dependent calcium channel (VDCC) blocker.
M9720 Aranidipine Aranidipine (MPC1304) is a calcium channel blocker which may positively affect ambulatory blood pressure. *This compound is unstable in solutions, freshly prepared is recommended.
M9600 2-Aminoethyl diphenylborinate (2-APB) 2-Aminoethyl diphenylborinate (2-APB) is a cell-permeable inhibitor of IP3R, and regulate IP3-induced calcium release.
M7796 Fluspirilene Fluspirilene is a non-competitive L-type calcium channel antagonist (IC50 = 0.03 μM) and a dopamine receptor antagonist.
M7778 Dantrolene sodium salt Inhibitor of Ca2+ release from sarcoplasmic reticulum; muscle relaxant.
M7409 Thapsigargin Thapsigargin is a potent inhibitor of SERCA ATPase.
M7346 T16Ainh - A01 T16Ainh - A01 is a Ca2+-activated Cl- channel transmembrane protein 16A (TMEM16A) inhibitor.
M6092 Mirogabalin Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS.
M5922 Ranolazine Ranolazine is a calcium uptake inhibitor via the sodium/calcium channel, used to treat chronic angina.
M5756 L-Phenylalanine L-Phenylalanine is an antagonist at α2δ calcium channels with a Ki of 980 nM.
M5738 Levosimendan Levosimendan is a calcium sensitizer acting through calcium-dependent binding to cardiac troponin C (cTnC), provides treatment for heart failure.
M5733 Lercanidipine Lercanidipine hydrochloride is a calcium channel blocker of the dihydropyridine class.
M5723 Lacidipine Lacidipine is a L-type calcium channel blocker, used for treating high blood pressure.
M5717 Isradipine Isradipine is a potent and selective L-type voltage-gated calcium channel blocker, used to treat high blood pressure.
M5654 Flunarizine 2HCl Flunarizine 2HCl is a dihydrochloride salt form which is a calcium channel blocker with a Ki of 68 nM.
M5640 Fendiline HCl Fendiline is a nonselective calcium channel blocker.
M5629 Ethosuximide Ethosuximide is a succinimide anticonvulsant, used mainly in absence seizures; A calcium channel blocker.
M5607 Efonidipine hydrochloride monoethanolate Efonidipine(NZ-105) Hcl monoethanolate is a dual T-type and L-type calcium channel blocker (CCB).
M5550 Dantrolene sodium hemiheptahydrate Dantrolene sodium hemiheptahydrate ia a skeletal muscle relaxant that acts by interfering with excitation-contraction coupling in the muscle fiber.
M5538 Cromolyn sodium Cromolyn sodium is an antiallergic drug.
M5411 Amlodipine Besylate Amlodipine Besylate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
M5205 ML204 ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.
M5139 Amlodipine Amlodipine is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
M5080 Efonidipine hydrochloride Efonidipine Hcl is a dual T-type and L-type calcium channel blocker .
M5077 (S)-(-)-BAY K 8644 (S)-(-)-BAY K 8644 is a Ca2+ channel activator; L-type Ca2+ channel activator.
M5075 GV-58 GV-58 is a potent, selective N- and P/Q-type Ca2(addition) channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2(addition) channel; 20-fold less potent CDK inhibitor activity.
M5073 (R)-(+)-BAY K 8644 (R)-(+)-BAY K 8644 is a calcium channel inhibitor, inhibits Ba2+ currents (IBa) with IC50 of 975 nM.
M3959 Felodipine Felodipine is a L-type Ca2+ channel blocker that is selective over N-, R-, P/Q- and T-type channels with IC50 of 0.15 nM.
M3807 Ionomycin (Calcium salt) Ionomycin is a calcium ionophor and an antibiotic produced by Streptomyces conglobatus.
M3621 Ionomycin Ionomycin is a calcium ionophor and an antibiotic produced by Streptomyces conglobatus.
M3613 NP118809 NP-118809 (39-1B4) is a potent N-type calcium channel blockers (IC50= 0.11 uM) ; good selectivity over L-type calcium channels.
M3599 Pregabalin Pregabalin (Lyrica) is a 3-isobutyl derivative of gamma-amino butyric acid (GABA) with anti-convulsant, anti-epileptic, anxiolytic, and analgesic activities.
M3572 Manidipine Manidipine is a lipophilic, third-generation, highly vasoselective dihydropyridine calcium antagonist with an IC50 of 2.6 nM.
M3498 Nimodipine Nimodipine is a dihydropyridine derivative and an analogue of the calcium channel blocker nifedipine, with antihypertensive activity.Nimodipine decreases intracellular free Ca2+,Beclin-1 and autophagy.
M3462 Nisoldipine Nisoldipine (Sular) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.
M3455 Nitrendipine Nitrendipine is a dihydropyridine calcium channel blocker with an IC50 of 95 nM.
M3440 Nilvadipine Nilvadipine is a potent calcium channel blocker with an IC50 of 0.03 nM.
M3424 Nifedipine Nifedipine (BAY-a-1040) is a potent vasodilator agent with calcium antagonistic action.
M3365 Tetracaine hydrochloride Tetracaine hydrochloride is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor.
M3317 Acetylcholine Chloride The chemical compound Acetylcholine Chloride is a neurotransmitter in both the peripheral nervous system (PNS) and central nervous system (CNS) in many organisms including humans.
M3296 Manidipine dihydrochloride Manidipine dihydrochloride is a hydrochloride salt form of Manidipine, which is a calcium channel blocker with IC50 of 2.6 nM, used clinically as an antihypertensive. Phase 4.
M3210 Benidipine hydrochloride Benidipine hydrochloride is a hydrochloride salt form of benidipine which is a dihydropyridine calcium channel blocker.
M3118 Verapamil hydrochloride Verapamil hydrochloride is an L-type calcium channel blocker that is a class IV anti-arrhythmia agent.
M2820 Lomerizine dihydrochloride Lomerizine dihydrochloride is a relatively new L- and T-type calcium channel blocker used in the treatment of migraine.
M2425 Azelnidipine Azelnidipine is a novel dihydropyridine derivative, a L-type calcium channel blocker, and an antihypertensive.
M2257 Levetiracetam Levetiracetam (UCB L059) is an antiepileptic, it is also a selective M2 muscarinic acetylcholine receptors (mAChR) inhibitor.
M2248 Cilnidipine Cilnidipine is a dual L- and N-type calcium channel blocker that displays antihypertensive, sympatholytic and neuroprotective activity.
M1927 KB-R7943 mesylate KB-R7943 mesylate is a potent, selective inhibitor of the reverse mode of the Na+/Ca2+ exchanger (IC50 = 0.7 mM).

Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.