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  Catalog
Abmole Inhibitor Catalog 2017

Androgen Receptor Androgen Receptor

Inhibitors

Cat.No.  Name Information
M5586 DL-Epinephrine DL-Epinephrine(DL-Adrenaline) is a hormone and a neurotransmitter.
M5565 Dexmedetomidine HCl Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties.
M5544 Cyproterone Acetate Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity.
M5454 Betaxolol HCl Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM.
M5396 Alfuzosin HCl Alfuzosin HCl is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH).
M5395 Alfuzosin Alfuzosin is an α1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH).
M5035 17 alpha-propionate 17 alpha-propionate is a new topical and peripherally selective androgen antagonist.
M3750 TAK-700 TAK-700 (Orteronel) is an investigational, oral, nonsteroidal, selective, reversible inhibitor of 17,20-lyase, a key enzyme in the production of androgenic hormones.
M3685 Mesterolone The Mesterolone is an orally applicable androgen, and DHT derivative.
M3234 (R)-Bicalutamide (R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells.
M3191 Nilutamide Nilutamide (RU 23908) is an androgen receptor (AR) blocker with IC50 of 0.4 μM.
M3028 Spironolactone Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM.
M2717 Galeterone Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth.
M2670 Epiandrosterone Epiandrosterone is a steroid hormone with weak androgenic activity, is a natural metabolite of DHEA.
M2344 RU 58841 RU 58841 is a specific androgen receptor antagonist or anti-androgen.
M2270 ARN-509 ARN-509 is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC).
M2092 AZD3514 AZD3514 is a potent, small-molecule androgen receptor downregulator with potential anticancer cancer activity.
M1986 Andarine Andarine (GTx-007, S-4) is an orally active partial agonist for androgen receptors.
M1973 Ostarine Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM.
M1960 Bicalutamide Bicalutamide is an orally active non-steroidal androgen receptor antagonist (IC50 = 190 nM).


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