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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M8955 | MIN-101 | MIN-101 (Roluperidone) is a novel compound with affinities for 5-HT2A and sigma-2 receptors with Ki values of 7.53 nM and 8.19 nM, respectively. |
| M8942 | GSK163090 | GSK163090 is a potent, selective, and orally active 5-HT1A/B/D receptor antagonist. |
| M8932 | Eptapirone | Eptapirone (F11440) is a potent 5HT(1A) receptor agonist with marked anxiolytic and antidepressant potential. |
| M8900 | TG6-10-1 | TG6-10-1 is a potent and selective antagonist for the prostaglandin E2 receptor subtype EP2. |
| M8856 | WAY-100135 dihydrochloride | WAY-100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). |
| M6065 | Ziprasidone HCl monohydrate | Ziprasidone(CP88059) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. |
| M6064 | Ziprasidone HCl | Ziprasidone HCl is a novel and potent dopamine and serotonin (5-HT) receptor antagonist, used in the treatment of schizophrenia and bipolar disorder. |
| M6058 | Vortioxetine | Vortioxetine (Lu AA21004) is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively. |
| M6051 | Venlafaxine | Venlafaxine is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI) class. |
| M6050 | Venlafaxine HCl | Venlafaxine HCl is an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), used to treat major depressive disorder (MDD), generalised anxiety disorder (GAD), panic disorder and social phobia. |
| M6027 | Trazodone | Trazodone HCl is an antidepressant belonging to the class of serotonin receptor antagonists and reuptake inhibitors for treatment of anxiety disorders. |
| M5992 | Tegaserod maleate | Tegaserod maleate is a partial agonist of the 5-HT4 receptor; stimulates the peristaltic reflex and accelerates gastrointestinal transit. |
| M5989 | Tandospirone | Tandospirone(SM-3997) is a potent and selective 5-HT1A receptor partial agonist (Ki = 27 nM) that displays selectivity over SR-2, SR-1C, α1, α2, D1 and D2 receptors (Ki values ranging from 1300-41000 nM). |
| M5951 | Sarpogrelate HCl | Sarpogrelate(MCI-9042) hydrochloride, a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. |
| M5938 | Rizatriptan Benzoate | Rizatriptan Benzoate is an agonist at serotonin 5-HT1B and 5-HT1D receptors, used to treat acute migraine attacks. |
| M5935 | Risperidone | Risperidone is a mutil-targeted antagonist for dopamine, serotonin, adrenergic and histamine receptors, used to treat schizophrenia and bipolar disorder. |
| M5920 | Ramosetron HCl | Ramosetron Hydrochloride(YM060 Hydrochloride) is a serotonin 5-HT3 receptor antagonist for the treatment of nausea and vomiting. |
| M5884 | Pizotifen | Pizotifen(Pizotyline) is a highly selective 5-HT receptor blocking agent, which is a benzocycloheptane based drug. |
| M5861 | Paroxetine HCl | Paroxetine HCl is an antidepressant drug of the SSRI type. |
| M5835 | Ondansetron Hydrochloride Dihydrate | Ondansetron is a highly specific and selective serotonin 5-HT3 receptor antagonist (Ki=6.16 nM), with low affinity for dopamine receptors. |
| M5804 | Naftidrofuryl oxalate | Naftidrofuryl is a drug used in the management of peripheral and cerebral vascular disorders as a vasodilator, enhance cellular oxidative capacity, and may also be a 5-HT2 receptor antagonist. |
| M5799 | Mosapride Citrate | Mosapride Citrate is a gastroprokinetic agent that acts as a selective 5HT4 agonist. |
| M5798 | Mosapride | Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist. |
| M5754 | Loxapine | Loxapine Succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. |
| M5660 | Fluvoxamine maleate | Fluvoxamine Maleate is a selective serotonin (5-HT) reuptake inhibitor (SSRI), used in the treatment of obsessive-compulsive disorder. |
| M5548 | Dalasetron Mesylate hydrate | Dolasetron(MDL-73147) is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. |
| M5543 | Cyproheptadine hydrochloride sesquihydrate | Cyproheptadine hydrochloride sesquihydrate is an antihistamine and is an antagonist of serotonin and histamine2. |
| M5542 | Cyproheptadine HCl | Cyproheptadine is a histamine receptor antagonist for 5-HT2 receptor with IC50 of 0.6 nM. |
| M5475 | Cabergoline | Cabergoline, an ergot derivative, is a potent dopamine receptor agonist on D2 receptors. |
| M5466 | Blonanserin | Blonanserin is a relatively selective serotonin (5-HT)2A and dopamine D2 antagonist, used the treatment of schizophrenia. |
| M5424 | Asenapine maleate | Asenapine maleate is a high-affinity antagonist of serotonin, norepinephrine, dopamine and histamine receptors, used for the treatment of schizophrenia and acute mania associated with bipolar disorder. |
| M5423 | Asenapine | Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. |
| M5400 | Alosetron | Alosetron Hydrochloride is the hydrochloride salt form of alosetron, a potent and selective 5-HT3 receptor antagonist. |
| M5214 | Lasmiditan | Lasmiditan (also known as COL-144 and LY573144) is a high-affinity, highly selective serotonin (5-HT) 5-HT(1F) receptor agonist. |
| M5130 | Cisapride | Cisapride(R 51619) is a nonselective 5-HT4 receptor agonist, it is also a potent hERG potassium channel inhibitor. IC50 Value is 0.14 μM (EC50 for 5-HT4 receptor). |
| M5045 | Tianeptine | Tianeptine is a selective facilitator of 5-HT uptake in vitro and in vivo. |
| M5044 | Tianeptine sodium salt | Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo. |
| M5022 | Almotriptan Malate | Almotriptan Malate is a 5-HT1B/1D-receptor agonist used to treat migraine. |
| M3985 | Triptolide | Triptolide is a structurally unique diterpene triepoxide isolated from a traditional Chinese medicinal plant with anti-inflammatory, immunosuppressive, contraceptive and antitumor activities. |
| M3909 | Glycyrrhizic acid | Glycyrrhizic acid is a widely used anti-inflammatory agent isolated from the licorice root. |
| M3793 | Deferitrin | Deferitrin is a novel, orally available iron chelator, is in the early stage of clinical development for the treatment of chronic iron overload due to transfusional therapy. |
| M3791 | YM 90K hydrochloride | YM 90K hydrochloride is a selective AMPA antagonist with neuro-protective effect. AMPA is a transmembrane glutamate receptor composed of the subunits GluR-1,2,3,4. |
| M3790 | Tasosartan | Tasosartan is a selective, potent, orally active and long-acting nonpeptide Angiotensin II type 1 (AT1) receptor antagonist. |
| M3782 | Oxiracetam | Oxiracetam could decrease neural injury and increase ability of learning, memory and space cognition in traumatic brain injury rats. |
| M3772 | SB242084 | SB242084 has a high affinity (pKi 9.0) for the cloned human 5-HT2C receptor and 100- and 158-fold selectivity over the closely related cloned human 5-HT2B and 5-HT2A subtypes respectively. |
| M3748 | Mestanolone | Mestanolone is the 17α-methylated version of dihydrotestosterone (DHT). |
| M3659 | Pimavanserin | Pimavanserin is a selective serotonin 5-HT2A inverse agonist. |
| M3646 | Cyclobenzaprine hydrochloride | Cyclobenzaprine hydrochloride is a skeletal muscle relaxant and a central nervous system (CNS) depressant. |
| M3585 | Tropisetron | Tropisetron is a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist with an IC50 of 70.1 ± 0.9 nM for 5-HT3 receptor. |
| M3583 | Urapidil hydrochloride | Urapidil hydrochloride is an α1-adrenoceptor antagonist and 5-HT1A receptor agonist with pIC50 of 6.13 and 6.4 respectively. |
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