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Abmole Inhibitor Catalog 2017

OX Receptor OX Receptor


Cat.No.  Name Information
M9943 OXA (17-33) OXA (17-33) is a potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively).
M9855 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist (ABM-565520) is a potent and selective Orexin2 receptor agonist with EC50 value of 23 nM.
M9839 Lemborexant Lemborexant (E-2006) is an orally active, competitive and reversible dual OX1 and OX2 receptors antagonist, with IC50 values of 6.1 nM and 2.6 nM, respectively.
M9573 Orexin A (human, mouse, rat, bovine) Orexin A (human, mouse, rat, bovine) is a specific, high-affinity agonist for G-protein-coupled receptor OX1R.
M8997 MK-1064 MK-1064 is a potent, selective and orally active Orexin OX2 Receptor Antagonist for the research of insomnia.
M8966 SB-649868 SB-649868 is a selective orally active orexin (OX) receptor antagonist with pKi values of 9.4 and 9.5 at the OX1 and OX2 receptor, respectively.
M3796 SB-334867 hydrochloride SB-334867 hydrochloride is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
M3760 TCS-1102 TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively).
M3710 MK-3697 MK-3697 is an isonicotinamide small molecule, acting as a potent and selective Orexin 2 receptor antagonist with Ki = 0.95 nM.
M3324 SB408124 SB408124 (Tocris-1963) is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.
M2272 Suvorexant Suvorexant (MK-4305) is a potent, selective and orally bioavailable antagonist of OX(1)R and OX(2)R for the treatment of insomnia.
M2124 MK-6096 MK-6096 is an orally bioavailable potent and selective reversible antagonist of OX(1)R and OX(2)R.
M1711 Febuxostat Febuxostat (Uloric) is a non-purine selective xanthine oxidase inhibitor with IC50 of 114 -210 nM.

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