Free shipping on all orders over $ 500
  Catalog
Abmole Inhibitor Catalog 2017

OX Receptor OX Receptor

Inhibitors

Cat.No.  Name Information
M3796 SB-334867 SB-334867 is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
M3760 TCS-1102 TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively).
M3710 MK-3697 MK-3697 is an isonicotinamide small molecule, acting as a potent and selective Orexin 2 receptor antagonist with Ki = 0.95 nM.
M3324 SB408124 SB408124 (Tocris-1963) is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.
M2272 Suvorexant Suvorexant (MK-4305) is a potent, selective and orally bioavailable antagonist of OX(1)R and OX(2)R for the treatment of insomnia.
M2124 MK-6096 MK-6096 is an orally bioavailable potent and selective reversible antagonist of OX(1)R and OX(2)R.
M1711 Febuxostat Febuxostat (Uloric) is a non-purine selective xanthine oxidase inhibitor with IC50 of 114 -210 nM.


Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2017 AbMole BioScience. All Rights Reserved.