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OX Receptor Orexin Receptor

Cat.No.  Name Information
M9573 Orexin A (human, mouse, rat, bovine) Orexin A (human, mouse, rat, bovine) is a specific, high-affinity agonist for G-protein-coupled receptor OX1R.
M3261 Almorexant Almorexant is a competitive OX1 and OX2 orexin receptor antagonist with IC50 of 13 and 8 nM, respectively.
M40751 Daridorexant hydrochloride Daridorexant hydrochloride is an orally active dual orexin type 1 and type 2 (OX1 and OX2) receptor antagonist (DORA) as well as an inhibitor of BCRP, with an IC50 value of 3.0 μM when acting on BCRP, and can be used in studies related to insomnia.
M25479 [Ala11,D-Leu15]-Orexin B (human) acetate [Ala11,D-Leu15]-Orexin B (human) acetate is a potent and selective orexin-2 receptor (OX2) agonist. [Ala11,D-Leu15]-Orexin B (human) acetate shows a 400-fold selectivity for the OX2 (EC50=0.13 nM) over OX1 (EC50=52 nM).
M25478 Orexin B, human TFA Orexin B, human TFA is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.
M25477 Orexin B, rat, mouse TFA Orexin B, rat, mouse TFA is an endogenous orexin receptor agonist. Orexin B, rat, mouse TFA binds and activates two closely related orphan G protein-coupled receptors OX1-R and OX2-R.
M14036 Orexin A (human, rat, mouse) (TFA) Orexin A human, rat, mouse TFA, a 33 amino acid excitatory neuropeptide, orchestrates diverse central and peripheral processes.
M14035 EMPA EMPA is a high-affinity, reversible and selective orexin OX2 receptor antagonist. [3H]EMPA binds to human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM respectively.
M14034 Almorexant hydrochloride Almorexant hydrochloride (ACT 078573 hydrochloride) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM, respectively.
M10955 Daridorexant Daridorexant is an effective orexin receptor antagonist. It also has IC50s of 2 nM and 3 nM for the Ox1 receptor and Ox2 receptor, respectively.
M9943 OXA (17-33) OXA (17-33) is a potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively).
M9855 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist (ABM-565520) is a potent and selective Orexin2 receptor agonist with EC50 value of 23 nM.
M9839 Lemborexant Lemborexant (E-2006) is an orally active, competitive and reversible dual OX1 and OX2 receptors antagonist, with IC50 values of 6.1 nM and 2.6 nM, respectively.
M8997 MK-1064 MK-1064 is a potent, selective and orally active Orexin OX2 Receptor Antagonist for the research of insomnia.
M8966 SB-649868 SB-649868 is a selective orally active orexin (OX) receptor antagonist with pKi values of 9.4 and 9.5 at the OX1 and OX2 receptor, respectively.
M7396 TCS-OX2-29 TCS-OX2-29 is a potent, high affinities and selective orexin-2 receptor (OX2R) antagonist with an IC50 value of 40 nM and a pKI value of 7.5. TCS-OX2-29 displays ~250-fold selectivity for OX2 over OX1.
M7263 SB 334867 SB 334867 is a selective non-peptide OX 1 antagonist.
M6833 IPSU IPSU is a oX 2 receptor antagonist; orally bioavailable.
M3796 SB-334867 hydrochloride SB-334867 hydrochloride is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
M3760 TCS-1102 TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively).




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