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Abmole Inhibitor Catalog 2017

Opioid Receptor Opioid Receptor


Cat.No.  Name Information
M10432 Difelikefalin (CR-845; FE-202845) TFA Difelikefalin (CR-845; FE-202845) TFA is a peripherally restricted and selective agonist of kappa opioid receptor (KOR).
M10240 CTOP TFA CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively.
M10229 Porcine dynorphin A (1-13) Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist.
M9784 Naloxegol oxalate Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
M9615 DAMGO DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR.
M9514 JDTic JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects.
M9268 Met-Enkephalin Met-Enkephalin (H-Tyr-Gly-Gly-Phe-Met-OH) inhibits tumor growth via binding to the opioid receptor.
M6036 Trimebutine maleate Trimebutine maleate is a drug with antimuscarinic and weak mu opioid agonist effects.
M6035 Trimebutine Trimebutine is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain.
M5589 Docusate Sodium Docusate Sodium is a laxative used to treat constipation, for constipation due to the use of opiates it maybe used with a stimulant laxative, can be taken by mouth or rectally.
M5403 Alvimopan dihydrate Alvimopan dihydrate(LY 246736; ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery.
M5289 PZM21 PZM21 is a potent and selective μ-opioid-receptor (μOR) agonist with an EC50 of 1.8 nM.
M5067 Eluxadoline Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist.
M5065 Cebranopadol Cebranopadol is a novel first in class compounds with potent agonist activity on ORL-1 (opioid receptor like -1) and the well established mu opioid receptor.
M4808 TRV130 hydrochloride TRV130 hydrochloride (Oliceridine) is a novel μ-opioid receptor (MOR) G protein-biased ligand.
M3582 Racecadotril Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM
M2991 SA 4503 SA 4503 is a novel and selective opioid sigma1 receptor agonist with IC50 of 17.4 nM.
M2876 Naloxone hydrochloride Naloxone hydrochloride is an opioid inverse agonist compound used to counter the effects of opiate overdose.
M2214 JTC-801 JTC-801 is a novel opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM.
M2145 Loperamide hydrochloride Loperamide hydrochloride is a high affinity μ-opioid receptor agonist with peripheral selectivity with Ki values of 2, 48 and 1156 nM for μ-, δ- and κ-opioid receptors respectively.
M1953 ADL5859 Hydrochloride ADL5859 is a potent, selective and orally bioavailable δ-opioid receptor agonist (Ki = 0.84 nM, EC50 = 20 nM).
M1577 Naltrexone Hydrochloride Naltrexone hydrochlorideis an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence.

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