Free shipping on all orders over $ 500
Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M4808 | TRV130 hydrochloride | TRV130 hydrochloride (Oliceridine) is a novel μ-opioid receptor (MOR) G protein-biased ligand. |
| M14033 | Ro 64-6198 | Ro 64-6198 is a potent, selective, nonpeptide, high-affinity, high cellular permeability and brain penetration N/OFQ receptor (NOP) agonist with an EC50 value of 25.6 nM. |
| M14032 | Norbinaltorphimine dihydrochloride | Norbinaltorphimine dihydrochloride is a potent and selective κ opioid receptor antagonist. |
| M14031 | Methylnaltrexone Bromide | Methylnaltrexone Bromide, a quaternary derivative of Naltrexone, is an orally active and selective mu-opioid receptor antagonist, functions as a peripherally acting receptor antagonist in tissues of the gastrointestinal tract. |
| M14030 | Matrine | Matrine (Matridin-15-one) is an alkaloid found in plants from the Sophora genus. It has a variety of pharmacological effects, including anti-cancer effects, and action as a kappa opioid receptor and u-receptor agonist. |
| M14029 | Aticaprant | Aticaprant (CERC-501) is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. |
| M14028 | Deltorphin 2 TFA | Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor. |
| M11311 | BMS-986122 | Bms-986122 is a selective and effective positive allosteric regulator of μ -opioid receptor (µ-OR). Bms-986122 showed enhancement of β -inhibitory protein recruitment, adenylate cyclase inhibition and G-protein activation mediated by normal agonists. Bms-986122 enhances damGO-mediated [35S]GTPγS binding in mouse meninges. |
| M11163 | Dermorphin | Dermorphin is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin. Dermorphin can be used to suppress neuralgia. |
| M10584 | SR17018 | SR17018 is an mu-opioid-receptor (MOR) agonist, EC50 is 97 nM for binding with GTPγS. |
| M10570 | Adrenorphin (Metorphamide) | Adrenorphin (Metorphamide) is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM. |
| M10564 | CYT-1010 | CYT-1010 is a mu-opioid receptor agonist with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. |
| M10563 | Dynorphin A (1-8) | Dynorphin A (1-8) is the most likely natural ligand of the kappa receptor. Dynorphin A (1-8) inhibited 3H-Bremazocine binding to the purified kappa receptor with IC50 of 303 nM. |
| M10510 | LY2940094 | LY-2940094 is a potent, selective and orally available antagonist of nociceptin receptor (NOP receptor) with Ki of 0.105 nM and Kb of 0.166 nM. |
| M10484 | Nalfurafine hydrochloride | Nalfurafine hydrochloride (TRK-820 hydrochloride) is a potent selective and orally active kappa opioid receptor (KOR) agonist. |
| M10432 | Difelikefalin (CR-845; FE-202845) TFA | Difelikefalin (CR-845; FE-202845) TFA is a peripherally restricted and selective agonist of kappa opioid receptor (KOR). |
| M10240 | CTOP TFA | CTOP TFA is a peptide that acts as a potent and selective μ opioid receptor antagonist, with Ki values of 0.96 and >10,000 nM for μ and δ receptors, respectively. |
| M10229 | Porcine dynorphin A (1-13) | Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist. |
| M9784 | Naloxegol oxalate | Naloxegol oxalate (NKTR-118 oxalate; AZ-13337019 oxalate) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation. |
| M9615 | DAMGO | DAMGO is an opioid receptor agonist with the ability to affect the locomotive activity in rodents, Kd value is 3.46 nM for native μ-OPR. |
| M9514 | JDTic | JDTic is a kappa opioid receptor (KOR) antagonist that prevents stress-induced reinstatement of cocaine-maintained responding and has antidepressant-like effects. |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.
