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Abmole Inhibitor Catalog 2017

Cannabinoid Cannabinoid


Cat.No.  Name Information
M10218 (+)-Gallocatechin (+)-Gallocatechin is found notably in green tea, it has moderate affinity to the human cannabinoid receptor and acts as an antioxidant.
M9691 JD-5037 JD-5037 is a cannabinoid-1 receptor blocker (CB1R antagonist) with IC50 of 1.5 nM.
M9687 JWH-133 JWH-133 is a synthetic cannabinoid.
M9652 CB1-IN-1 CB1-IN-1 is a novel potent restricted CB1R antagonist with Ki of 0.3 nM and 21 nM for CB1R and CB2R, respectively.
M9136 Cannabidiol Cannabidiol is a GPR55 and weak CB1 antagonist with IC50s of 0.445 and 3.35 μM, it is also a CB2 receptor inverse agonist and inhibitor of anandamide uptake with IC50 of 27.5 μM.
M8985 LY2828360 LY2828360 is a novel potent, selective, and efficacious CB2 cannabinoid agonist.
M8919 BAY 59-3074 BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively.
M7325 Rimonabant Hydrochloride Rimonabant hydrochloride is a cannabinoid receptor antagonist, which binds selectively to central cannabinoid receptors (CB1) with high affinity
M6429 AM 630 AM 630 is a CB2 selective inverse agonist.
M5290 (±)-SLV-319 (±)-SLV319 (Ibipinabant) is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo.
M3282 GW842166X GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.
M3266 WIN 55212-2 mesylate WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively.
M2981 Rimonabant Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
M2552 CP 945598 CP 945598 (Otenabant) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
M2461 BML-190 BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.
M2343 AM-2201 AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.
M2051 CP 945598 hydrochloride CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively).
M2012 AM1241 AM1241 is a cannabinoid CB2 receptor selective agonist.
M1907 Org 27569 Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor.

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