Catalog

Cannabinoid Cannabinoid

Inhibitors

Cat.No.	Name	Information
M4845	CP945598	CP945598 HCl is a potent and selective cannabinoid receptor CB1 antagonist with Ki of 0.7 nM, exhibits 10,000-fold greater selectivity against human CB2 receptor.
M3282	GW842166X	GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.
M3266	WIN 55212-2 mesylate	WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively.
M2552	CP 945598	CP 945598 (Otenabant) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
M2461	BML-190	BML-190 is a selective cannabinoid CB2 receptor inverse agonist with K_i of 435 nM, with 50-fold selectivity over CB1 receptor.
M2343	AM-2201	AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.
M2051	CP 945598 hydrochloride	CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively).
M2012	AM1241	AM1241 is a cannabinoid CB2 receptor selective agonist.
M1907	Org 27569	Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor.