|M8985||LY2828360||LY2828360 is a novel potent, selective, and efficacious CB2 cannabinoid agonist.|
|M8919||BAY 59-3074||BAY-59-3074 is a novel cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively.|
|M5290||(±)-SLV-319||(±)-SLV319 (Ibipinabant) is a potent and selective CB1 receptor antagonist (Ki = 7.8 nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo.|
|M3282||GW842166X||GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor.|
|M3266||WIN 55212-2 mesylate||WIN 55212-2 is a potent nanomolar affinity cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM at the human cloned CB1 and CB2 receptors respectively.|
|M2981||Rimonabant||Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.|
|M2552||CP 945598||CP 945598 (Otenabant) is a selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.|
|M2461||BML-190||BML-190 is a selective cannabinoid CB2 receptor inverse agonist with Ki of 435 nM, with 50-fold selectivity over CB1 receptor.|
|M2343||AM-2201||AM-2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.|
|M2051||CP 945598 hydrochloride||CP 945598 hydrochloride is a selective and high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively).|
|M2012||AM1241||AM1241 is a cannabinoid CB2 receptor selective agonist.|
|M1907||Org 27569||Org 27569 is a potent and selective allosteric modulator of the cannabinoid CB1 receptor.|
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