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Vernakalant

Cat. No. M3622

All AbMole products are for research use only, cannot be used for human consumption.

Vernakalant Structure
Synonym:

RSD-1235

Size Price Availability
10mg USD 375  USD375 Out of stock
50mg USD 960  USD960 Out of stock
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Quality Control & Documentation
Biological Activity

Vernakalant (RSD-1235) is an investigational mixed ion channel blocker that can terminate acute atrial fibrillation (AF) in humans at 2 to 5 mg/kg and may be more atrial-selective than available agents; in treatment of antiarrhythmic. Vernakalant is shown to have good conversion rates, an apparently safe antiarrhythmic profile and is well tolerated in patients with a history of ischemic heart disease.

Chemical Information
Molecular Weight 349.47
Formula C20H31NO4
CAS Number 794466-70-9
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Blomström-Lundqvist C, et al. Expert Opin Drug Saf. Safety and efficacy of pharmacological cardioversion of atrial fibrillation using intravenous vernakalant, a new antiarrhythmic drug with atrial selectivity.

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Keywords: Vernakalant, RSD-1235 supplier, Potassium Channel, inhibitors, activators

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