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Methoxyphenamine HCl

Cat. No. M5781
Methoxyphenamine HCl Structure
Size Price Availability Quantity
50mg USD 80 In stock
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Quality Control
  • Current batch:
  • Purity >98%
  • COA
  • MSDS
Biological Activity

Methoxyphenamine Hydrochloride is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 215.72
Formula C11H18ClNO
CAS Number 5588-10-3
Purity >98%
Solubility 34 mg/mL in DMSO
Storage at -20°C
References

Methoxyphenamine inhibits basal and histamine-induced nasal congestion in anaesthetized rats.
Lau WA, et al. Br J Pharmacol. 1990 Oct;101(2):394-8. PMID: 1701679.

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  Catalog
Abmole Inhibitor Catalog 2017




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