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GMQ hydrochloride

Cat. No. M6755

All AbMole products are for research use only, cannot be used for human consumption.

GMQ hydrochloride Structure
Size Price Availability Quantity
10mg USD 55  USD55 In stock
50mg USD 110  USD110 In stock
100mg USD 185  USD185 In stock
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Quality Control & Documentation
Biological Activity

GMQ hydrochloride is a selective opener of acid-sensing ion channel 3 (ASIC3) at pH 7.4. GMQ hydrochloride alters the pH dependence of ASIC1a and ASIC1b. GMQ hydrochloride does not affect the activation curve of ASIC2a. GMQ can be used for the research of neurological disease.

Chemical Information
Molecular Weight 237.69
Formula C10H11N5.HCl
CAS Number 5361-15-9
Form Solid
Solubility (25°C) DMSO 2 mg/mL
Water 3 mg/mL
Storage 4°C, protect from light, dry, sealed
References

[1] Lauth, et al. Proc Natl Acad Sci. Inhibition of GLI-mediated transcription and tumor cell growth by small-molecule antagonists.

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Keywords: GMQ hydrochloride supplier, Sodium Channel, inhibitors, activators

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