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GLPG2938

Cat. No. M21147

All AbMole products are for research use only, cannot be used for human consumption.

GLPG2938  Structure

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Quality Control & Documentation
Biological Activity

GLPG2938 is a potent and selective S1P2 antagonist.GLPG2938 can be used in the study of idiopathic pulmonary fibrosis (IPF).

Chemical Information
Molecular Weight 503.40
Formula C20H19F6N7O2
CAS Number 2130996-00-6
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Oscar Mammoliti, et al. J Med Chem. Discovery of the S1P2 Antagonist GLPG2938 (1-[2-Ethoxy-6-(trifluoromethyl)-4-pyridyl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea), a Preclinical Candidate for the Treatment of Idiopathic Pulmonary Fibrosis

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  Catalog
Abmole Inhibitor Catalog




Keywords: GLPG2938 supplier, LPL Receptor, inhibitors, activators

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