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Ethisterone

Cat. No. M5628

Ethisterone Structure
Size Price Availability Quantity
100mg USD 75 In stock
500mg USD 115 In stock
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Quality Control
  • Current batch:
  • Purity >99%
  • COA
  • MSDS
Biological Activity

Ethisterone is a progestogen hormone being considered to treat prostate cancer.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 312.45
Formula C21H28O2
CAS Number 434-03-7
Purity >99%
Solubility 0.05 mg/mL in DMSO
Storage at -20°C
References

Click chemistry inspired highly facile synthesis of triazolyl ethisterone glycoconjugates.
Kumar D, et al. Steroids. 2014 Feb;80:71-9. PMID: 24316164.

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  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Ethisterone supplier, Estrogen Receptor, inhibitors

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