All AbMole products are for research use only, cannot be used for human consumption.
Endoxifen is the key active metabolite of Tamoxifen and an estrogen receptor (ER) modulator with high affinity and specificity for the estrogen receptor and inhibits aromatase activity.Endoxifen has been used in studies related to breast cancer, sclerofibroblastoma, and bipolar disorder.
| Molecular Weight | 373.49 |
| Formula | C25H27NO2 |
| CAS Number | 110025-28-0 |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[5] V Craig Jordan. J Clin Oncol. Endoxifen: The End, or Are We at the Beginning?
| Related Estrogen Receptor Products |
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| Idoxifene
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| (R)-Equol
(R)-Equol is an agonist of both ERα and ERβ with Kis of 27.4 and 15.4 nM, respectively. |
| (Rac)-Vepdegestrant
(Rac)-Vepdegestrant is the isomer of Vepdegestrant. |
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