Free shipping on all orders over $ 500

Desogestrel

Cat. No. M5564
Desogestrel Structure
Synonym:

Cerazette, Desogen, Desogestrelum, Org-2969

Size Price Availability Quantity
10mg USD 70 In stock
50mg USD 150 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control
  • Current batch:
  • Purity >98%
  • COA
  • MSDS
Biological Activity

Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 310.47
Formula C22H30O
CAS Number 54024-22-5
Purity >98%
Solubility 62 mg/mL in DMSO
Storage at -20°C
References

Desogestrel versus danazol as preoperative treatment for hysteroscopic surgery: a prospective, randomized evaluation.
Laganà AS, et al. Gynecol Endocrinol. 2014 Nov;30(11):794-7. PMID: 24919887.

Related Estrogen Receptor Products
Relugolix

Relugolix, also known as TAK-385, is a luteinizing hormone-releasing hormone (LH-RH) receptor antagonist with an IC50 of 0.12 nM.

Elagolix sodium

Elagolix Soidum is a potent, selective, orally active, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with Kd value of 54 pM.

GDC-0810

GDC-0810 (Brilanestrant, ARN-81) is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM.

Tamoxifen

Tamoxifen is a estrogen receptor partial agonist/antagonist.

GSK 4716

GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.

  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Desogestrel, Cerazette, Desogen, Desogestrelum, Org-2969 supplier, Estrogen Receptor, inhibitors

Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2017 AbMole BioScience. All Rights Reserved.