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BAY 1214784

Cat. No. M21311

All AbMole products are for research use only, cannot be used for human consumption.

BAY 1214784  Structure

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Quality Control & Documentation
Biological Activity

BAY 1214784 is a potent, selective and orally active antagonist of the human gonadotropin-releasing hormone receptor (hGnRH-R).BAY 1214784 has the potential to be studied in uterine fibroids.

Chemical Information
Molecular Weight 672.11
Formula C29H26ClF4N3O5S2
CAS Number 1631164-25-4
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Olaf Panknin, et al. J Med Chem. Discovery and Characterization of BAY 1214784, an Orally Available Spiroindoline Derivative Acting as a Potent and Selective Antagonist of the Human Gonadotropin-Releasing Hormone Receptor as Proven in a First-In-Human Study in Postmenopausal Women

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Keywords: BAY 1214784 supplier, inhibitors, activators

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