|M9242||ISRIB||ISRIB is a potent and selective PERK inhibitor with IC50 of 5 nM.|
|M7425||trans-ISRIB||trans-ISRIB is a integrated stress response (ISR) inhibitor.|
|M2996||Salubrinal||Salubrinal is a selective inhibitor of eIF2α dephosphorylation and inhibits ER stress-mediated apoptosis with EC50 of ~15 μM.|
|M2735||GSK2656157||GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM, 500-fold greater against a panel of 300 kinases.|
|M2734||GSK2606414||GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM, displaying at least 100-fold selectivity over the other EIF2AKs assayed.|
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.