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Neurokinin Receptor Neurokinin Receptor

Cat.No.  Name Information
M40803 Pavinetant Pavinetant is a neurokinin-3 receptor (NK3R) antagonist that may be used in studies related to hot flashes and polycystic ovary syndrome.
M31366 Elinzanetant Elinzanetant (NT-814) is a first-in-class, orally active dual neurokinin receptor NK1/NK3 antagonist for studies related to hot flushes (HFs).
M30886 Rolapitant hydrochloride hydrate Rolapitant hydrochloride hydrate (SCH619734 hydrochloride hydrate) is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a Ki of 0.66 nM. Rolapitant hydrochloride hydrate does not interact with CYP3A4. Rolapitant hydrochloride hydrate shows potent anti-emetic activity in a ferret emesis model.
M27671 Vapreotide Vapreotide is a neurokinin-1 (NK1) receptor antagonist, with an IC50 of 330 nM.
M25564 Substance P (6-11) Substance P (6-11) is the C-terminal hexapeptideamide of Substance P. Substance P (6-11) binds to NK-1 tachykinin receptor. Substance P (6-11) shows depolarization of motoneurons and a hypotensive effect.
M14024 Substance P TFA Substance P TFA (Neurokinin P TFA) is a neuropeptide, acting as a neurotransmitter and as a neuromodulator in the CNS. The endogenous receptor for substance P is neurokinin 1 receptor (NK1-receptor, NK1R).
M14021 Fezolinetant Fezolinetant is an antagonist of the neurokinin 3 receptor (NK3R), used for the treatment of menopausal hot flushes.
M10332 Vapreotide acetate Vapreotide acetate (BMY-41606 acetate; RC160 acetate) is a neurokinin-1 (NK1) receptor antagonist with IC50 value of 330 nM.
M9080 Substance P Substance P is a neuropeptide, acting as a neurotransmitter and as a neuromodulator.The endogenous receptor for substance P is neurokinin 1 receptor (NK1-receptor, NK1R).
M9019 Rolapitant Rolapitant (SCH619734) is an orally bioavailable, centrally-acting, selective neurokinin 1 receptor (NK1-receptor) antagonist with a Ki of 0.66 nM.
M7735 CP-96345 CP-96345 is a highly potent and selective, orally active tachykinin and substance P receptor non-peptide inhibitor.
M7258 SB 223412 SB 223412 is a potent, selective non-peptide NK3 antagonist. Brain penetrant.
M3882 Netupitant Netupitant is a selective neurokinin 1 (NK1) receptor antagonist with potential antiemetic activity with Ki of 0.95 nM.
M2712 Fosaprepitant dimeglumine salt Fosaprepitant is a water-soluble phosphoryl procompound for Aprepitant which is a NK1 antagonist.*The compound is unstable in solutions, freshly prepared is recommended
M2673 Eprazinone dihydrochloride Eprazinone is a mucolytic.
M1832 Maropitant Maropitant (Cerenia) is a novel, selective neurokinin type-1 (NK1) receptor antagonist.
M1650 Aprepitant Aprepitant (Emend) is an antiemetic chemical compound that belongs to a class of compounds called substance P antagonists (SPA).
M1569 Monohydroxy Netupitant Monohydroxy Netupitant is the metabolite of Netupitant, which is a highly selective NK1 receptor antagonist.
M54512 Spantide II Spantide II, an undecapeptide substance P (SP) analog, is a potent neurokinin-1 receptor (NK-1R) antagonist.
M54402 Substance P (7-11) Substance P (7-11) is a C-terminal fragment of Substance P which can cause an increase in the intracellular calcium concentration.




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