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Neurokinin Receptor Neurokinin Receptor

Inhibitors

Cat.No.  Name Information
M14024 Substance P TFA Substance P TFA (Neurokinin P TFA) is a neuropeptide, acting as a neurotransmitter and as a neuromodulator in the CNS. The endogenous receptor for substance P is neurokinin 1 receptor (NK1-receptor, NK1R).
M14023 NKP608 NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective, specific and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50=2.6 nM) and in vivo.
M14022 Neurokinin A TFA Neurokinin A TFA (Substance K TFA), a peptide neurotransmitter of the tachykinin family, acts via the NK-2 receptor. Neurokinin A acts as a major mediator in human airway and gastrointestinal tissues.
M14021 Fezolinetant Fezolinetant is an antagonist of the neurokinin 3 receptor (NK3R), used for the treatment of menopausal hot flushes.
M10342 [Leu31,Pro34]-NPY TFA (human,rat) [Leu31,Pro34]-NPY TFA (human,rat) is a specific neuropeptide Y1 receptor agonist.
M10332 Vapreotide acetate Vapreotide acetate (BMY-41606 acetate; RC160 acetate) is a neurokinin-1 (NK1) receptor antagonist with IC50 value of 330 nM.
M9200 Ibodutant Ibodutant (MEN15596) is a potent and selective tachykinin NK2 receptor antagonist with a pKi of 10.1.
M9185 Serlopitant Serlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist.
M9080 Substance P Substance P is a neuropeptide, acting as a neurotransmitter and as a neuromodulator.The endogenous receptor for substance P is neurokinin 1 receptor (NK1-receptor, NK1R).
M9019 SCH 619734 SCH-619734 is an orally bioavailable, centrally-acting, selective neurokinin 1 receptor (NK1-receptor) antagonist with a Ki of 0.66 nM.
M7258 SB 223412 SB 223412 is a potent, selective non-peptide NK3 antagonist. Brain penetrant.
M6303 JNJ-31020028 JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat); >100-fold selective versus human Y1/Y4/Y5 receptors.
M3882 Netupitant Netupitant is a selective neurokinin 1 (NK1) receptor antagonist with potential antiemetic activity with Ki of 0.95 nM.
M1832 Maropitant Maropitant (Cerenia) is a novel, selective neurokinin type-1 (NK1) receptor antagonist.
M1650 Aprepitant Aprepitant (Emend) is an antiemetic chemical compound that belongs to a class of compounds called substance P antagonists (SPA).



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