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Abmole Inhibitor Catalog 2017

Histamine Receptor Histamine Receptor

Inhibitors

Cat.No.  Name Information
M5458 Bilastine Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria.
M5393 Alcaftadine Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines. Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor.
M3665 Promethazine hydrochloride Promethazine hydrochloride is a potent histamine H1 receptor antagonist, used as a sedative and antiallergic medication.
M3487 Azelastine hydrochloride Azelastine hydrochloride is a potent, second-generation, selective, histamine antagonist.
M3458 Chlorpheniramine Maleate Chlorpheniramine (Chlorpheniramine maleate, Chlorphenamine) is an histamine H1 receptor antagonist with IC50 of 12 nM.
M3454 Olopatadine hydrochloride Olopatadine hydrochloride is a histamine blocker and mast cell stabilizer with an IC50 of 559 μM for the release of histamine.
M3431 Nizatidine Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.
M3385 Cimetidine Cimetidine, a histamine congener, competitively inhibits histamine binding to histamine H2 receptors.
M3318 Clemastine Fumarate Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM.
M3226 Brompheniramine hydrogen maleate Brompheniramine hydrogen maleate is a histamine H1 receptors antagonist.
M3091 Tripelennamine hydrochloride Tripelennamine is a widely used H1 antagonist, inhibiting PhIP glucuronidation with IC50 of 30 μM.
M2990 Rupatadine Fumarate Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
M2919 Pemirolast potassium Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.
M2811 Levodropropizine Levodropropizine possess anti-allergic and inhibits histamine receptor, reduces cough by interfering with stimulus activation of peripheral endings of sensory nerves and by modulation of neuropeptides involved in the cough reflex.
M2784 JNJ-7777120 JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM, exhibits >1000-fold selectivity over the other histamin receptors.
M2760 Hydroxyzine dihydrochloride Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM.
M2756 Histamine dihydrochloride Histamine is an organic nitrogen compound, acts on target cells in mammalian brain via stimulation of Histamine 1/2.
M2699 Fexofenadine hydrochloride Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
M2660 Ebastine Ebastinea is a potent H1-histamine receptor antagonist, used for allergic disorders.
M2650 Doxepin hydrochloride Doxepin is a psychotropic agent with tricyclic antidepressant and anxiolytic properties.
M2621 Desloratadine Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
M2582 Clemizole Clemizole is a H1 histamine receptor antagonist with IC50 Value of 8 mM (NS4B).
M2545 Cyclizine dihydrochloride Cyclizine 2HCl is a piperazine derivative with Histamine H1 receptor antagonist activity.
M2522 Ciproxifan Ciproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
M2477 Buclizine hydrochloride Buclizine hydrochloride is an antihistamine and anticholinergic of the piperazine derivative family.
M2452 Betahistine dihydrochloride Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.
M2449 Bepotastine Besilate Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
M2416 Azatadine dimaleate Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
M2088 Ciproxifan maleate Ciproxifan is an orally bioavailable, extremely potent histamine H3 inverse agonist/antagonist.


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