|M10818||FT827||FT827 is a selective covalent inhibitor of ubiquitin-specific protease 7 (USP7) (Ki=4.2 µM)。 FT827 with USP7 Catalytic Domain (USP7CDresidues 208-560) combined, apparent Kd The value is 7.8 μM.|
|M10817||FT671||FT671 is a potent, non-covalent, selective USP7 inhibitor,IC50 The value is 52 nM, bound to the USP7 catalytic domain Kd The value is 65 nM.|
|M10753||VLX1570||VLX1570 is a competitive inhibitor of proteasome deuteronase (DUBs),IC50 约10 μM。|
|M10752||GNE-6776||GNE-6776 is a potent, selective USP7 inhibitor with oral activity.|
|M10504||IU1-47||IU1-47 is a potent and specific USP14 inhibitor with an IC50 of 0.6 μM.|
|M9871||GSK2643943A||GSK2643943A is a deubiquitylating enzyme (DUB) inhibitor targeting USP20/Ub-Rho with an IC50 of 160 nM.|
|M9785||ML364||ML364 is a small molecule inhibitor of the deubiquitinase USP2 (IC50=1.1 μM) with potential anticancer activity.|
|M9654||GRL0617||GRL0617 is a potent, selective and competitive noncovalent inhibitor of SARS PLPro, with IC50 of 0.6 μM and Ki of 0.49 μM.|
|M9639||SJB2-043||SJB2-043 is an inhibitor of USP1 which targets ID1 degradation in leukemic cells.|
|M2807||LDN-57444||LDN-57444 is a reversible, competitive proteasome inhibitor for Uch-L1 with IC50 of 0.88 μM, 28-fold selectivity over isoform Uch-L3.|
|M2565||PR-619||PR-619 is a non-selective, reversible inhibitor of the deubiquitinylating enzymes (DUBs) with EC50 of 1-20 μM.|
|M2431||b-AP15||b-AP15 is a deubiquitinases inhibitor for 19S proteasomes activity of Ub-AMC cleavage with IC50 of 2.1 μM. *The compound is unstable in solutions, freshly prepared is recommended|
|M2196||P22077||P22077 is a selective inhibitor of ubiquitin-specific protease (USP) 7 with EC50 of 8.6 μM.|
|M2195||P5091||P5091 is a potent and selective inhibitor of ubiquitin-specific protease (USP) 7 with IC50 of 4.2 μM.|
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.