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Ozagrel sodium

Cat. No. M5847

Ozagrel sodium Structure
Size Price Availability Quantity
10mg USD 75 In stock
50mg USD 200 In stock
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Quality Control
  • Current batch:
  • Purity >99%
  • COA
  • MSDS
Biological Activity

Ozagrel(OKY-046) sodium salt is an antiplatelet agent working as a thromboxane A2 synthesis inhibitor.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 250.23
Formula C13H11N2NaO2
CAS Number 130952-46-4
Purity >99%
Solubility 44 mg/mL in water
Storage at -20°C
References

Preischemic neuroprotective effect of minocycline and sodium ozagrel on transient cerebral ischemic rat model.
Park SI, et al. Brain Res. 2015 Mar 2;1599:85-92. PMID: 25555371.

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  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Ozagrel sodium supplier, Factor Xa, inhibitors

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