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Nelfinavir Mesylate

Cat. No. M3654
Nelfinavir Mesylate Structure


Size Price Availability Quantity
10mM*1mL In DMSO USD 88 In stock
5mg USD 60 In stock
10mg USD 90 In stock
50mg USD 240 In stock
100mg USD 440 In stock
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Quality Control
  • Current batch:
  • Purity >98%
  • COA
  • MSDS
Biological Activity

Nelfinavir Mesylate (also known as AG1343) is a potent enzyme inhibitor (Ki = 2 nM) and antiviral agent (HIV-1 ED50 = 14 nM). Nelfinavir (AG1343) is well absorbed orally in a variety of species and possesses favorable pharmacokinetic properties in humans. AG1343 (Viracept) has recently been approved for marketing for the treatment of AIDS.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 663.89
Formula C33H49N3O7S2
CAS Number 159989-65-8
Purity >98%
Solubility DMSO: ≥ 20 mg/mL
Storage at -20°C

Viracept (nelfinavir mesylate, AG1343): a potent, orally bioavailable inhibitor of HIV-1 protease.
Kaldor SW, et al. J Med Chem. 1997 Nov 21;40(24):3979-85. PMID: 9397180.

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Keywords: Nelfinavir Mesylate, AG-1343 supplier, HIV Protease, inhibitors

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