| Cat.No. | Name | Information |
|---|---|---|
| M3480 | Tolvaptan | Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM for the inhibition of AVP-induced platelet aggregation. |
| M11395 | Lixivaptan | Lixivaptan (VPA-985, WAY-VPA 985) is an orally active, selective vasopressin receptor V2 antagonist with IC50 values of 1.2 nM in humans and 2.3 nM in rats. |
| M5166 | Conivaptan hydrochloride | Conivaptan hydrochloride is a non-peptide vasopressin receptor antagonist, which can inhibit V1A receptor in rat liver and V2 receptor in kidney with Ki values of 0.48 and 3.04 nM, respectively. |
| M52877 | Big Endothelin-1 (1-39), porcine | Big Endothelin-1 (1-39), porcine is the precursor of endothelin-1. |
| M52876 | D[LEU4, LYS8]-VP | D[LEU4,LYS8]-VP is a selective agonist of vasopressin V1b receptor, with the Kis of 0.16 nM, 0.52 nM, and 0.1.38 nM for rat, human and mouse V1b receptor, respectively. |
| M52875 | (D-Arg8)-Inotocin | (D-Arg8)-Inotocin is a potent, selective and competitive antagonist of vasopressin receptor (V1aR), with a Ki of 1.3 nM. |
| M52874 | [Deamino-Pen1, Val4, D-Arg8]-vasopressin | [Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an arginine-vasopressin (AVP) antagonist. |
| M52873 | [8-L-arginine] deaminovasopressin | [8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog. |
| M52872 | (Phe2, Orn8)-Oxytocin | (Phe2,Orn8)-Oxytocin is a selective V1 vasopressin agonist. |
| M52871 | (d(CH2)51, Tyr(Me)2, Dab5, Arg8)-Vasopressin | (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71. |
| M52870 | Desamino(D-3-(3′-pyridyl)-Ala2, Arg8)-Vasopressin | Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), is a weak agonist at antidiuretic receptor. |
| M52869 | (Phenylac1, D-Tyr(Et)2, Lys6, Arg8, des-Gly9)-Vasopressin | (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist. |
| M52868 | 2-(3-Trifluoromethylphenyl)glycine hydrochloride | 2-(3-Trifluoromethylphenyl)glycine hydrochloride is a precursor of substituted 2-acetamido-5-aryl-l, 2,4-triazolones. |
| M52867 | Dp[Tyr(methyl)2, Arg8]-Vasopressin | Dp[Tyr(methyl)2,Arg8]-Vasopressin is a non-selective peptide arginine vasopressin Vlb receptor antagonist. |
| M52866 | Terlipressin acetate | Terlipressin acetate is a vasopressin analogue with potent vasoactive properties. |
| M52865 | Val9-Oxytocin | Val9-Oxytocin is a full antagonist of vasopressin (V1a) receptor. |
| M52864 | JKC 301 | JKC 301 is a selective Endothelin A receptor antagonist. |
| M52863 | F992 | F992 is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue. |
| M41952 | Invopressin | Invopressin is a vasopressin V1A receptor partial agonist (EC50: 1.0 nM). |
| M31222 | SKF 100398 | SKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP. |
| M31042 | Selepressin acetate | Selepressin (FE 202158) acetate is a selective vasopressin V1A receptor agonist. Selepressin is a potent vasopressor. Selepressin can be used in the research of septic shock. |
| M30785 | Selepressin | Selepressin (FE 202158) is a selective vasopressin V1A receptor agonist. Selepressin is a potent vasopressor. Selepressin can be used in the research of septic shock. |
| M30218 | SRX246 | SRX246 is a potent, CNS-penetrant, highly selective, orally bioavailable vasopressin 1a (V1a) receptor antagonist (Ki=0.3 nM for human V1a). SRX246 has no interaction at V1b and V2 receptors. SRX246 also displays negligible binding at 64 others receptors classes, including 35 G-proteincoupled receptors. SRX246 can be used for treatment of stress-related disorders. |
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