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Abmole Inhibitor Catalog 2017

GABA Receptor GABA Receptor

Inhibitors

Cat.No.  Name Information
M9114 LAU159 LAU159 is a potent, functionally selective α6β3γ2 GABAA receptor modulator.
M8879 AOA hemihydrochloride Aminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T.
M6010 Tiagabine HCl Tiagabine Hydrochloride is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
M6009 Tiagabine Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
M5870 Pentylenetetrazol Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist.
M5730 L-Cycloserine L-cycloserine irreversibly inhibit GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals in a time-dependent manner, results in increased levels of gamma-aminobutyric acid (GABA), which is an inhibitory neurotransmitter in vivo.
M5669 Gabapentin HCl Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
M5653 Flumazenil Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.
M5575 Dihydroergotoxine mesylate Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site.
M5442 Baclofen Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.
M5390 Afloqualone Afloqualone is a agonist of GABA receptor .
M5378 Acamprosate calcium Acamprosate calcium (Campral EC) is a GABA receptor agonist and glutamate system modulator.
M4815 Vigabatrin Vigabatrin is a selective GABA-T (transaminase) inhibitor.
M3981 Bilobalide Bilobalide, a natural product extracted from Ginkgo biloba leaf, is known to exhibit a number of pharmacological activities.
M3968 Dihydromyricetin Dihydromyricetin is a natural antioxidant flavonoid from Ampelopsis grossedentata.
M3938 Baicalin Baicalin is a known prolyl endopeptidase inhibitor that induces apoptosis in pancreatic cancer cells.
M3600 Gabapentin Gabapentin is a pharmaceutical agent, specifically a GABA analogue.
M3344 Nefiracetam Nefiracetam is a GABAergic, cholinergic, and monoaminergic neuronal systems enhancer for Ro 5-4864-induced convulsions.
M2555 AWD 131-138 AWD 131-138 is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models.
M2347 (+)-Bicuculline (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.
M2005 (R)-Baclofen (R)-baclofen is a selective gamma-aminobutyric acid(B) agonist.
M1893 Etomidate Etomidate (marketed as Amidate) is a general anesthetic with GABA modulatory and GABA-mimetic actions.
M1891 SKF 89976A hydrochloride SKF 89976A hydrochloride is a potent GABA uptake inhibitor, selective for GAT-1.


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