Catalog

GABA Receptor GABA Receptor

Inhibitors

Cat.No.	Name	Information
M6066	Zolpidem	Zolpidem is a benzodiazepine agonist with high selectivity for α1-subunit-containing GABAA receptors.
M6010	Tiagabine HCl	Tiagabine Hydrochloride is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
M6009	Tiagabine	Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor.
M5880	Piperazine	Piperazine, GABA receptor agonist, is an anthelmintic used in the treatment of the intestinal nematodes Ascaris lumbricoides and Enterobius vermicularis.
M5870	Pentylenetetrazol	Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist.
M5730	L-Cycloserine	L-cycloserine irreversibly inhibit GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals in a time-dependent manner, results in increased levels of gamma-aminobutyric acid (GABA), which is an inhibitory neurotransmitter in vivo.
M5669	Gabapentin HCl	Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
M5668	Gabapentin	Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.
M5653	Flumazenil	Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses.
M5575	Dihydroergotoxine mesylate	Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site.
M5442	Baclofen	Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.
M5420	Armodafinil	Armodafinil is the R-enantiomer of the racemic synthetic agent modafinil with central nervous system (CNS) stimulant and wakefulness-promoting activities
M5390	Afloqualone	Afloqualone is a agonist of GABA receptor .
M5378	Acamprosate calcium	Acamprosate calcium (Campral EC) is a GABA receptor agonist and glutamate system modulator.
M3981	Bilobalide	Bilobalide, a natural product extracted from Ginkgo biloba leaf, is known to exhibit a number of pharmacological activities.
M3968	Dihydromyricetin	Dihydromyricetin is a natural antioxidant flavonoid from Ampelopsis grossedentata.
M3600	Gabapentin	Gabapentin is a pharmaceutical agent, specifically a GABA analogue.
M3344	Nefiracetam	Nefiracetam is a GABAergic, cholinergic, and monoaminergic neuronal systems enhancer for Ro 5-4864-induced convulsions.
M3167	Picrotoxinin	Picrotoxinin is a GABA_A receptor antagonist that binds to the GABA receptor-linked Cl⁻ channel.
M2555	AWD 131-138	AWD 131-138 is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models.
M2347	(+)-Bicuculline	(+)-Bicuculline is a competitive antagonist of GABA_A receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.
M2005	(R)-Baclofen	(R)-baclofen is a selective gamma-aminobutyric acid(B) agonist.
M1893	Etomidate	Etomidate (marketed as Amidate) is a general anesthetic with GABA modulatory and GABA-mimetic actions.
M1891	SKF 89976A hydrochloride	SKF 89976A hydrochloride is a potent GABA uptake inhibitor, selective for GAT-1.

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