Certificate of Analysis
| Product Name: | S1RA |
| Catalog Number: | M2596 |
| CAS Number: | 878141-96-9 |
Physical and Chemical Properties
| Formula: | C20H23N3O2 |
| Molecular Weight: | 337.42 |
| Solubility: | DMSO 30 mg/mL (ultrasonic and warming and heat to 60°C); 1M HCl : 40 mg/mL (ultrasonic and adjust pH to 1 with HCl) |
| Storage: |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Chemical Structure: |  |
Analytical Data
| QC Standard: | >98.0% |
| H-NMR: | Consistent with structure |
Product Information
| Description: | S1RA (E-52862) is a potent and selective sigma-1 receptor (σ1R, Ki=17 nM), which showes good selectivity against σ2R (Ki > 1000 nM). |
| Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |