Product Name: | Pulrodemstat benzenesulfonate |
Catalog Number: | M10727 |
CAS Number: | 2097523-60-7 |
Formula: | C30H29F2N5O5S |
Molecular Weight: | 609.65 |
Solubility: | DMSO ≥ 60 mg/mL |
Storage: | -20°C, dry, sealed |
Chemical Structure: | ![]() |
QC Standard: | >99% |
H-NMR: | Consistent with structure |
Description: | CC-90011 (Pulrodemstat) benzenesulfonate is a potent, selective, reversible and orally active lysine-specific demethylase-1 (LSD1) inhibitor,IC50 0.25 nM. CC-90011 benzenesulfonate has less enzymatic inhibition of LSD2, MOA-A and MAO-B. CC-90011 benzenesulfonate induces differentiation of acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells and has potent anti-cancer activity. |
Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |