Certificate of Analysis

 

Product Name: PF-CBP1 HCl
Catalog Number: M20613
CAS Number: 2070014-93-4

Physical and Chemical Properties
Formula: C29H37ClN4O3
Molecular Weight: 525.08
Solubility: DMSO 100 mg/mL; Water 100 mg/mL
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: PF-CBP1 HCl Structure
Analytical Data
QC Standard: >99%
H-NMR: Consistent with structure
Product Information
Description: PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.