Certificate of Analysis
| Product Name: | PDK4-IN-1 hydrochloride |
| Catalog Number: | M21648 |
| CAS Number: | 2310262-11-2 |
Physical and Chemical Properties
| Formula: | C22H20ClN3O2 |
| Molecular Weight: | 393.87 |
| Solubility: | DMSO ≥ 90 mg/mL |
| Storage: | 2-8°C, dry, sealed |
| Chemical Structure: |  |
Analytical Data
| QC Standard: | 99.68% |
| H-NMR: | Consistent with structure |
Product Information
| Description: | PDK4-IN-1 hydrochloride is an anthraquinone derivative and a potent and orally active pyruvate dehydrogenase kinase 4 (PDK4) inhibitor with an IC50 value of 84 nM. PDK4-IN-1 hydrochloride potently represses cellular transformation and cellular proliferation and induces apoptosis. |
| Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |