Certificate of Analysis

 

Product Name: (αR,8aS)-GSK1614343 
Catalog Number: M27777
CAS Number: 1092476-84-0

Physical and Chemical Properties
Formula: C22H23F6N5O
Molecular Weight: 487.44
Form: Solid
Storage: Powder -20°C
Chemical Structure: (αR,8aS)-GSK1614343  Structure
Analytical Data
QC Standard: ≥99.0%
H-NMR: Consistent with structure
Product Information
Description: (αR,8aS)-GSK1614343 (compound 18a, d2) is a cyclized ghrelin antagonist with an pIC50 value of 8.4. (αR,8aS)-GSK1614343 shows a competitive antagonism of hGHSR1a with a mean pKb value of 8.06.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.