Product Name: | PROTAC BET degrader-2 |
Catalog Number: | M14874 |
CAS Number: | 2093388-33-9 |
Molecular Weight: | 770.84 |
Solubility: | DMSO 50 mg/mL |
Storage: | -20°C, sealed |
Chemical Structure: | ![]() |
QC Standard: | >99% |
H-NMR: | Consistent with structure |
Description: | PROTAC BET degrader-2 is a PROTAC connected by ligands for Cereblon and BET with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression. |
Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |