Certificate of Analysis

 

Product Name: Olcegepant hydrochloride
Catalog Number: M13934
CAS Number: 586368-06-1

Physical and Chemical Properties
Molecular Weight: 906.11
Solubility: DMSO 90 mg/mL; Water ≥ 66.66 mg/mL
Storage: 2-8°C, sealed
Chemical Structure: Olcegepant hydrochloride Structure
Analytical Data
QC Standard: >99%
H-NMR: Consistent with structure
Product Information
Description: Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.