Certificate of Analysis
| Product Name: | J-2156 TFA |
| Catalog Number: | M29587 |
| CAS Number: | 2387505-73-7 |
Physical and Chemical Properties
| Formula: | C26H29F3N4O6S |
| Molecular Weight: | 582.59 |
| Form: | Solid |
| Solubility: | Water 100 mg/mL (ultrasonic); DMSO 100 mg/mL (ultrasonic) |
| Storage: | Store at ≤ -20°C, protect from light, dry, sealed |
| Chemical Structure: |  |
Analytical Data
| QC Standard: | ≥99.0% |
| H-NMR: | Consistent with structure |
Product Information
| Description: | J-2156 TFA is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. J-2156 TFA has anti-inflammatory activity and it is used for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws in rats. |
| Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |