Product Name: | GSK864 |
Catalog Number: | M8651 |
CAS Number: | 1816331-66-4 |
Formula: | C30H31FN6O4 |
Molecular Weight: | 558.6 |
Form: | Solid |
Solubility: | DMSO: 10 mg/mL |
Storage: |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
Chemical Structure: |
QC Standard: | 99.99% |
H-NMR: | Consistent with structure |
Description: | GSK864 is a cell penetrant, potent and selective allosteric inhibitor of isocitrate dehydrogenase 1 (IDH1) that potently inhibits intracellular 2-hydroxyglutarate (2-HG) production in HT-1080 cells. |
Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |