Certificate of Analysis

 

Product Name: GSK864
Catalog Number: M8651
CAS Number: 1816331-66-4

Physical and Chemical Properties
Formula: C30H31FN6O4
Molecular Weight: 558.6
Form: Solid
Solubility: DMSO: 10 mg/mL
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: GSK864 Structure
Analytical Data
QC Standard: 99.99%
H-NMR: Consistent with structure
Product Information
Description: GSK864 is a cell penetrant, potent and selective allosteric inhibitor of isocitrate dehydrogenase 1 (IDH1) that potently inhibits intracellular 2-hydroxyglutarate (2-HG) production in HT-1080 cells.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.