Product Name: | Gambogenic acid |
Catalog Number: | M11241 |
CAS Number: | 173932-75-7 |
Formula: | C38H46O8 |
Molecular Weight: | 630.78 |
Solubility: | DMSO ≥ 200 mg/mL |
Storage: | 4°C, protect from light, dry, sealed |
Chemical Structure: | ![]() |
QC Standard: | >99% |
H-NMR: | Consistent with structure |
Description: | Gambogenic acid is the active ingredient in Huangteng and has anti-cancer activity. Gambogenic acid is an effective EZH2 inhibitor, which specifically covalently binds to Cys668 in the EZH2-SET domain to induce EZH2 ubiquitination. |
Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |