Certificate of Analysis
| Product Name: | DRAK2-IN-1 |
| Catalog Number: | M49489 |
| CAS Number: | 871837-60-4 |
Physical and Chemical Properties
| Formula: | C21H20N4O3 |
| Molecular Weight: | 376.41 |
| Form: | Solid |
| Solubility: | DMSO 100 mg/mL |
| Storage: |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Chemical Structure: |  |
Analytical Data
| QC Standard: | >99.0% |
| H-NMR: | Consistent with structure |
Product Information
| Description: | DRAK2-IN-1 is a potent, selective, ATP-competitive DRAK2 inhibitor with IC50 and Ki values of 3 nM and 0.26 nM, respectively.In addition, DRAK2-IN-1 also inhibits DRAK1 (IC50=51 nM). |
| Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |