Certificate of Analysis

 

Product Name: CP-154526 hydrochloride
Catalog Number: M8038
CAS Number: 257639-98-8

Physical and Chemical Properties
Formula: C23H32N4 · HCl
Molecular Weight: 400.99
Solubility: DMSO: 10 mg/mL
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: CP-154526 hydrochloride Structure
Analytical Data
QC Standard: >98%
H-NMR: Consistent with structure
Product Information
Description: CP-154526 hydrochloride is a selective, non-peptide antagonist of corticotropin releasing factor receptors (CRF1) with a Ki of 2.7 nM. CP 154526 hydrochloride shows selective for CRF1 over CRF2 (Ki = >10 μM).
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.