Certificate of Analysis

 

Catalog Number: M2736
Product Name: GSK343
CAS Number: 1346704-33-3

Physical and Chemical Properties
Formula: C31H39N7O2
Molecular Weight: 541.69
Solubility: DMSO
Long-term Storage: at -20℃
Chemical Structure: GSK343 Structure
Analytical Data
HPLC: Shows Min >99% purity
H-NMR: Consistent with structure
Product Information
Description: GSK343 is a potent and selective EZH2 inhibitor with IC50 of 4 nM, showing 60 fold selectivity against EZH1, and >1000 fold selectivity against other histone methyltransferases.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials at -20°C or below and used within 1 month.