Certificate of Analysis


Catalog Number: M5259
Product Name: Citarinostat
CAS Number: 1316215-12-9

Physical and Chemical Properties
Formula: C24H26ClN5O3
Molecular Weight: 467.95
Solubility: 93 mg/mL in DMSO
Storage: at -20°C
Chemical Structure: Citarinostat Structure
Analytical Data
HPLC: Shows Min >98% purity
H-NMR: Consistent with structure
Product Information
Description: Citarinostat (ACY-241) is an orally available selective HDAC6 inhibitor with IC50 of 2.6 nM and 46 nM for HDAC6 and HDAC3, respectively. It has 13 to 18-fold selectivity towards HDAC6 in comparison to HDAC1-3.
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.