Certificate of Analysis

 

Catalog Number: M8923
Product Name: CCG215022
CAS Number: 1813527-81-9

Physical and Chemical Properties
Formula: C26H22FN7O3
Molecular Weight: 499.5
Solubility: DMSO: ≥ 10 mg/mL
Long-term Storage: at -20°C
Chemical Structure: CCG215022 Structure
Analytical Data
HPLC: Shows Min >98% purity
H-NMR: Consistent with structure
Product Information
Description: CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50 values of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, GRK5 and GRK1, respectively.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials at -20°C or below and used within 1 month.