Free shipping on all orders over $ 500

 About 33 results found for searched term "Aurora Kinase" (0.084 seconds)

Cat.No.  Name Target
M3931 Aurora Kinase Inhibitor III Aurora Kinase
Aurora Kinase Inhibitor 3
Aurora Kinase Inhibitor III is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM.
M29284 Aurora kinase inhibitor-8  Aurora Kinase
Aurora kinase inhibitor-8 is a highly selective inhibitor of the Aurora kinases.
M29927 Aurora kinase inhibitor-2  Aurora Kinase
Aurora kinase inhibitor-2 is a selective and ATP-competitive Aurora kinase inhibitor with IC50s of 310 nM and 240 nM for Aurora A and Aurora B, respectively.
M41412 Aurora Kinases-IN-4 Aurora Kinase
Aurora Kinases-IN-4 is a covalent and ATP competitive aurora kinase A inhibitor (IC50: 1.7 nM).
M1655 AT9283 Aurora Kinase
AT9283 is a potent inhibitor of several protein kinases, including Aurora A, Aurora B, Janus kinase 2 (JAK2), JAK3, and ABL.
M1691 CCT-129202 Aurora Kinase
CCT129202 is an Aurora kinase inhibitor with IC50 of 0.042 ± 0.022, 0.198 ± 0.05, and 0.227 ± 0.064 μmol/L for Aurora A, Aurora B, and Aurora C, respectively.
M1706 ENMD-2076 Aurora Kinase
ENMD-2076 is an orally-active, Aurora A/angiogenic kinase inhibitor.
M1752 MLN8237 (Alisertib) Aurora Kinase
Alisertib
MLN8237 (Alisertib) is a second-generation, orally bioavailable, highly selective Aurora kinase A inhibitor with IC50 of 61 nM.
M1769 PHA-739358 (Danusertib) Aurora Kinase
Danusertib
PHA-739358 (Danusertib) is a small molecule with low nanomolar activity against all aurora kinases (AKs) with IC50 value of 13 nM for aurora-A and 79 nM for aurora-B respectively.
M1800 JNJ-7706621 CDK
JNJ7706621
JNJ-7706621 is a dual cell cycle inhibitor with activity against cyclin-dependent kinases (CDK1, 2, 3, 6) with an IC50 of 3-175 nM and Aurora kinases (A and B) with an IC50 of 11-15 nM respectively.
M1815 KW-2449 FLT3
KW2449
KW-2449 is a novel multitargeted kinase inhibitor of FLT3, ABL and Aurora kinase with IC50 values of 6.6 nM, 14 nM and 48 nM.
M1877 ZM447439 Aurora Kinase
ZM-447439
ZM447439 is the first Aurora family kinase inhibitor with IC50 of 50 nM for Aurora B kinase.
M1881 Tozasertib Aurora Kinase
VX-680, MK-0457
Tozasertib (VX-680, MK-0457) is a potent and selective pan-Aurora kinase inhibitor active against all Bcr/Abl proteins.
M2103 CCT137690 Aurora Kinase
CCT137690 is a potent inhibitor of Aurora kinases with IC50 values of 15, 19 and 25 nM at Aurora A, Aurora C and Aurora B respectively.
M2127 Hesperadin Aurora Kinase
Hesperadin is an ATP-competitive inhibitor of Aurora B kinase with IC50 of 250 nM.
M2169 AMG 900 Aurora Kinase
AMG 900 is a potent and selective, orally available small molecule aurora kinase inhibitor.
M2188 Reversine Aurora Kinase
Reversine is a novel small molecule ATP-competitive Aurora kinase inhibitor with IC50 of 98.5 nM for Aurora B.
M5236 BI-847325 MEK
BI-847325 is an orally bioavailable, and selective dual MEK/Aurora kinase inhibitor with IC50 of 3 nM, 25 nM, 15 nM, 25 nM, and 4 nM for Xenopus laevis Aurora B, human Aurora A and Aurora C, as well as human MEK1 and MEK2, respectively.
M7363 TC-A 2317 hydrochloride Others
TC-A 2317 hydrochloride is a potent, selective Aurora kinase A inhibitor.
M7393 TC-S 7010 Others
TC-S 7010 is a potent and selective Aurora kinase A inhibitor.
M7986 OM137 Others
OM137 is an inhibitor of aurora kinases; inhibitor of spindle checkpoint.
M8042 CP-335963 Others
CP-335963 is an aurora 2 kinase inhibitor, PDGF inhibitor, and anti-proliferative.
M9895 LY3295668 Aurora Kinase
AK-01
LY3295668 (AK-01) is a potent, orally active and highly specific Aurora-A kinase inhibitor, with Ki values of 0.8 nM and 1038 nM for AurA and AurB, respectively.
M10945 Chiauranib VEGFR/PDGFR
CS2164
Chiauranib (CS2164) is a first-in-class orally active multi-target inhibitor of tumor angiogenesis.Chiauranib potently inhibits the angiogenesis-related kinases (VEGFR1, VEGFR2, VEGFR3, PDGFRα and c-Kit), mitosis-related kinase Aurora B and chronic inflammation-related kinase CSF-1R. Chiauranib has strong anticancer activity.
M13591 Cenisertib Aurora Kinase
AS-703569; R-763
Cenisertib (AS-703569) is an ATP-competitive multi-kinase inhibitor that blocks the activity of Aurora-kinase-A/B, ABL1, AKT, STAT5 and FLT3.
M20235 WAY-632963 Aurora Kinase
WAY-632963 is a Aurora kinase A inhibitor.
M20238 WAY-634704 Aurora Kinase
WAY-634704 is a Aurora kinase A inhibitor.
M20244 WAY-635764 Aurora Kinase
WAY-635764 is a Aurora kinase A inhibitor.
M20245 WAY-635767 Aurora Kinase
WAY-635767 is a Aurora kinase A inhibitor
M20246 WAY-636900 Aurora Kinase
WAY-636900 is a Aurora kinase A inhibitor.
M20247 WAY-636982 Aurora Kinase
WAY-636982 is a Aurora kinase A inhibitor.
M20251 WAY-638641 Aurora Kinase
WAY-638641 is a Aurora kinase A inhibitor.
M20284 WAY-661516 Aurora Kinase
WAY-661516 is a Aurora kinase A inhibitor.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2023 AbMole BioScience. All Rights Reserved.