Free shipping on all orders over $ 500

Regadenoson

Cat. No. M5924
Regadenoson Structure
Size Price Availability Quantity
5mg USD 90 In stock
10mg USD 155 In stock
50mg USD 420 In stock
Bulk Inquiry?

Quality Control
  • Current batch:
  • Purity >99%
  • COA
  • MSDS
Biological Activity

Regadenoson is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 390.35
Formula C15H18N8O5
CAS Number 313348-27-5
Purity >99%
Solubility 10 mM in DMSO
Storage at -20°C
References

Comparison of the Safety of Adenosine and Regadenoson in Patients Undergoing Outpatient Cardiac Stress Testing.
Brink HL, et al. Pharmacotherapy. 2015 Dec;35(12):1117-23. PMID: 26684552.

Related Adenosine Receptor Products
ZM241385

ZM-241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.

CGS 21680

CGS 21680 is a selective adenosine receptor agonist for A2A and A3 with Ki of 15 ng/mL and 37 ng/mL, respectively.

Istradefylline

Istradefylline is a selective adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM.

CGS 21680 hydrochloride

CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM.

SYN115

SYN115 is a novel, selective adenosine A(2A) receptor antagonist.

  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Regadenoson supplier, Adenosine Receptor, inhibitors

Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2017 AbMole BioScience. All Rights Reserved.