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Mestanolone

Cat. No. M3748
Mestanolone Structure
Size Price Availability Quantity
Free Sample (0.5-1 mg)  USD 0 In stock
100mg USD 60 In stock
500mg USD 120 In stock
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Quality Control
Biological Activity

Mestanolone is an orally bioavailable androgenic steroid that is highly androgenic while only slightly anabolic. It is incapable of aromatization and is not an agonist of the progesterone receptor. 17alpha-methyl-5alpha-androstan-3beta,16beta,17beta-triol is a very useful screening target for the doping test of MTS and Mestanolone in racehorses.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 304.48
Formula C20H32O2
CAS Number 521-11-9
Purity 99.92%
Solubility DMSO
Storage at -20°C
References

Identification and quantification of metabolites common to 17alpha-methyltestosterone and mestanolone in horse urine.
Yamada M, et al. J Pharm Biomed Anal. 2007 Sep 21;45(1):125-33. PMID: 17709226.

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