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Armodafinil

Cat. No. M5420
Armodafinil Structure
Synonym:

CEP-10953, CRL 40982, Armodafinil

Size Price Availability Quantity
10mg USD 90 In stock
50mg USD 325 In stock
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Quality Control
  • Current batch:
  • Purity >99%
  • COA
  • MSDS
Biological Activity

Armodafinil is the R-enantiomer of the racemic synthetic agent modafinil with central nervous system (CNS) stimulant and wakefulness-promoting activities

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of resveratrol used for a mouse (22.4 mg/kg) to a dose based on the BSA for a rat, multiply 22.4 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for resveratrol of 11.2 mg/kg.

Chemical Information
Molecular Weight 273.35
Formula C15H15NO2S
CAS Number 112111-43-0
Purity >99%
Solubility 54 mg/mL in DMSO
Storage at -20°C
References

Adjunctive armodafinil for major depressive episodes associated with bipolar I disorder.
Ketter TA, et al. J Affect Disord. 2015 Aug 1;181:87-91. PMID: 25933099.

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  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Armodafinil, CEP-10953, CRL 40982, Armodafinil supplier, GABA Receptor, inhibitors

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