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Alarelin Acetate

Cat. No. M5391
Alarelin Acetate Structure
Synonym:

Alarelin

Size Price Availability Quantity
5mg USD 65  USD65 In stock
10mg USD 105  USD105 In stock
50mg USD 150  USD150 In stock
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Quality Control & Documentation
Biological Activity

Alarelin acetate is a synthetic GnRH agonist. Alarelin is found in higher amounts than that of LH-RH in rat hypophyseal stimulation of gonadotropin secretion in vivo and in vitro and in ovulation inductions.

Chemical Information
Molecular Weight 1287.42
Formula C60H86N26O16
CAS Number 79561-22-1
Form Solid
Solubility (25°C) ≥ 58 mg/mL in DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Conversion of different model animals based on BSA (PMID: 27057123)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of Compound A used for a mouse (20 mg/kg) to a dose based on the BSA for a rat, multiply 20 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for Compound A of 10 mg/kg.

References

[1] Zhan Y, et al. J Chromatogr B Analyt Technol Biomed Life Sci. Rapid and sensitive liquid chromatography-tandem mass spectrometry method for the determination of leuprolide in human serum.

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