| Cat.No. | Name | Information |
|---|---|---|
| M11395 | Lixivaptan | Lixivaptan (VPA-985, WAY-VPA 985) is an orally active, selective vasopressin receptor V2 antagonist with IC50 values of 1.2 nM in humans and 2.3 nM in rats. |
| M5166 | Conivaptan hydrochloride | Conivaptan hydrochloride is a non-peptide vasopressin receptor antagonist, which can inhibit V1A receptor in rat liver and V2 receptor in kidney with Ki values of 0.48 and 3.04 nM, respectively. |
| M3480 | Tolvaptan | Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM for the inhibition of AVP-induced platelet aggregation. |
| M49895 | Felypressin acetate | Felypressin acetate is a non-catecholamine vasoconstrictor and an agonist of vasopressin 1. |
| M21942 | Balovaptan | Balovaptan (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. |
| M14067 | Argipressin | Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1. |
| M11457 | Desmopressin Acetate | Desmopressin is a synthetic octapeptide that is an analogue of the human hormone arginine vasopressin and has antidiuretic and procoagulant effects. |
| M11397 | D[LEU4,LYS8]-VP TFA | D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptors, with Ki values of 0.16 nM, 0.52 nM and 1.38 nM for rat, human and mouse V1b receptors, respectively. D[LEU4,LYS8]-VP TFA showed weak antidiuretic, vasopressor and oxytocin activity in vitro. |
| M11396 | Terlipressin diacetate | Terlipressin diacetate is a vasopressin analogue and a highly selective vasopressin V1 receptor agonist that reduces visceral blood flow and portal vein pressure and controls acute varicose rupture bleeding. Terlipressin diacetate has anti-inflammatory and antioxidant effects and can be used to study hepatorenal syndrome and norepinephrine-resistant septic shock. |
| M11394 | Felypressin | Felypressin (PLV-2) is a non-catecholamine vasoconstrictor and a vasopressin 1 (Vasopressin 1) agonist. Felypressin is widely used in dental surgery. |
| M11393 | RG7713 | RG7713 (RO5028442) is a highly effective and selective brain-osmotic vasopressin 1A (V1a) receptor antagonist with Ki values of 1 nM (hV1a) and 39 nM (mV1a). |
| M10312 | Argipressin Acetate | Argipressin (Arg8-vasopressin) binds to vascular arginine vasopressin receptors V1, V2 and V3, and its Kd value against V1 in A7r5 rat aortic smooth muscle cells is 1.31 nM. |
| M10242 | Antagonist G | Antagonist G is an anticancer peptide and it is also a potent vasopressin antagonist. |
| M6879 | L-371,257 | L-371,257 is a potent and selective oxytocin receptor antagonist. |
| M5431 | Atosiban Acetate | Atosiban (RW22164; Tractocile) Acetate is a nonapeptide, desamino-oxytocin analogue, and a competitive vasopressin/oxytocin receptor antagonist (VOTra). Atosiban inhibits the oxytocin-mediated release of inositol trisphosphate from the myometrial cell membrane. |
| M1917 | Mozavaptan | Mozavaptan (OPC-31260) is a selective vasopressin V2 receptor antagonist. |
| M54211 | d[Cha4]-AVP | d[Cha4]-AVP is a potent and selective vasopressin (AVP) V1b receptor agonist with a Ki of 1.2 nM for human V1b receptor. |
| M52880 | Big Endothelin-1 (1-38), human | Big Endothelin-1 (1-38), human is the precursor of endothelin-1. |
| M52879 | (d(CH2)51, Tyr(Me)2, Arg8)-Vasopressin | (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist. |
| M52878 | [Asu1, 6-Arg8]Vasopressin | [Asu1,6-Arg8]Vasopressin is an vasopressin agonist which potentiates cyclic AMP accumulation and ACTH release induced by corticotropin-releasing factor (CRF) in rat anterior pituitary cells in culture. |
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