| Cat.No. | Name | Information |
|---|---|---|
| M2358 | 3-Deazaneplanocin A | 3-deazaneplanocin A (DZNeP), an analog of adenosine, is a competitive inhibitor of S-adenosylhomocysteine hydrolase with Ki of 50 pM. |
| M4804 | GSK-503 | GSK-503 is a potent EZH2 inhibitor with potential anticancer activity. |
| M3631 | AZ505 | AZ505 ditrifluoroacetate is a potent and highly selective inhibitor of the oncogenic protein SMYD2 (IC50=0.12 uM) with potential anticancer activity. |
| M3105 | UNC0646 | UNC0646 is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP with IC50 of 6 nM and 15 nM , respectively, with excellent potency in a variety of cell lines and excellent separation of functional potency versus cell toxicity. |
| M3103 | UNC0631 | UNC0631 is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP with IC50 of 6 nM and 15 nM, respectively, with excellent potency in a variety of cell lines and excellent separation of functional potency versus cell toxicity. |
| M3101 | UNC0224 | UNC0224 is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP with IC50 of 15 nM and 20 nM, respectively. |
| M2861 | MM-102 | MM-102 is a high-affinity peptidomimetic MLL1 inhibitor with IC50 of 0.4 μM. |
| M2675 | EPZ004777 hydrochloride | EPZ004777 hydrochloride is the hydrochloride salt of EPZ004777, which is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM. |
| M2334 | EPZ004777 | EPZ004777 is a potent, selective, small-molecule inhibitor of DOT1L with IC50 of 0.4 nM. |
| M2179 | EPZ-5676 | EPZ-5676 is a potent and selective aminonucleoside inhibitor of DOT1L histone methyltransferase. |
| M2024 | BIX 01294 Trihydrochloride | BIX 01294 Trihydrochloride is a potent inhitor of G9a histone methyltransferase with IC50 of 2.7 μM. |
| M53317 | SAH-EZH2 | SAH-EZH2, a stable EZH2 α-helical peptide, is an EZH2/EED interaction inhibitor. |
| M53316 | UNC4976 | UNC4976 is a positive allosteric modulator (PAM) peptidomimetic of CBX7 chromodomain binding to nucleic acids. |
| M53315 | C21 | C21 is a potent, irreversible, and selective PRMT1 inhibitor with an IC50 of 1.8 μM. |
| M41699 | EZH2-IN-15 | EZH2-IN-15 (SHR2554) is a EZH2 inhibitor. |
| M41698 | NSD-IN-2 | NSD-IN-2 is a potent and irreversible NSD1 inhibitor. |
| M41697 | MS9715 | MS9715 is a potent and seletive NSD3-targeting PROTAC. |
| M41696 | NSD2-IN-4 | NSD2-IN-4 is a potent and selective NSD2-SET inhibitor. |
| M41695 | PRMT4-IN-1 | PRMT4-IN-1 is a selective inhibitor of PRMT4 (IC50=3.2 nM). |
| M41694 | WM-662 | WM-662 is a WDR5-MYC interaction inhibitor, with an IC50 of 18 μM. |
| M41693 | PRMT5-IN-25 | PRMT5-IN-25 is a potent PRMT5 inhibitor with an Ki value of 0.06 nM. |
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